Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 824
TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293397BDBM293397(US10106522, Example 1)
Affinity DataIC50: 25nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293403BDBM293403(US10106522, Example 3)
Affinity DataIC50: 28nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293407BDBM293407(US10106522, Example 5)
Affinity DataIC50: 54nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293406BDBM293406(US10106522, Example 4)
Affinity DataIC50: 93nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293400BDBM293400(US10106522, Example 2)
Affinity DataIC50: 115nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293409BDBM293409(US10106522, Example 8)
Affinity DataIC50: 169nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293408BDBM293408(US10106522, Example 7)
Affinity DataIC50: 175nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293410BDBM293410(US10106522, Example 9)
Affinity DataIC50: 195nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293414BDBM293414(US10106522, Compound I-11 in CN 103896915)
Affinity DataIC50: 260nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293413BDBM293413(US10106522, Compound I-3 in CN 103896915)
Affinity DataIC50: 271nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293411BDBM293411(US10106522, Example 5 in EP 0580541)
Affinity DataIC50: 424nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent

TargetHistamine H1 receptor(Human)
Faes Farma

US Patent
LigandChemical structure of BindingDB Monomer ID 293412BDBM293412(US10106522, Compound I-8 in CN 103896915)
Affinity DataIC50: 1.99E+3nMpH: 7.4 T: 2°CAssay Description:Affinity for histamine H1-receptor was determined by binding studies to H1 receptors. The sample used is a suspension of membranes of CHO cells trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2019
Entry Details
US Patent