Compile Data Set for Download or QSAR
Report error Found 144 Enz. Inhib. hit(s) with all data for entry = 50038480
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50188578BDBM50188578(8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376936BDBM50376936(CHEMBL408266)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50188547BDBM50188547(8-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-diethyl...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376954BDBM50376954(CHEMBL259342)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376955BDBM50376955(CHEMBL260490)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376948BDBM50376948(CHEMBL259300)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376944BDBM50376944(CHEMBL258499)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376952BDBM50376952(CHEMBL258507)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376949BDBM50376949(CHEMBL259524)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50188583BDBM50188583(8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376953BDBM50376953(CHEMBL260976)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50233082BDBM50233082(8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322845BDBM50322845(3-methyl-1-propyl-8-(1-(3-(trifluoromethyl)benzyl)...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50233076BDBM50233076(8-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-dipropy...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376938BDBM50376938(CHEMBL428086)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376940BDBM50376940(CHEMBL427736)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376942BDBM50376942(CHEMBL259772)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376969BDBM50376969(CHEMBL258686)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376941BDBM50376941(CHEMBL259565)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376947BDBM50376947(CHEMBL412747)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376951BDBM50376951(CHEMBL409852)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322843BDBM50322843(8-(1-(3-(trifluoromethyl)benzyl)-1-pyrazol-4-yl)-1...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236738BDBM50236738(3-ethyl-1-propyl-8-(1-(3-(trifluoromethyl)benzyl)-...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322846BDBM50322846(3-ethyl-1-propyl-8-(1-((pyridin-3-yl)methyl)-1H-py...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376939BDBM50376939(CHEMBL410021)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376937BDBM50376937(CHEMBL407969)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376967BDBM50376967(CHEMBL427911)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376962BDBM50376962(CHEMBL408936)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236760BDBM50236760(8-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1,3-dimethy...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376968BDBM50376968(CHEMBL260763)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376945BDBM50376945(CHEMBL261819)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376964BDBM50376964(CHEMBL265212)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376946BDBM50376946(CHEMBL265213)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376948BDBM50376948(CHEMBL259300)
Affinity DataKi:  35nMAssay Description:Displacement of [125I]ABMECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376963BDBM50376963(CHEMBL430050)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376966BDBM50376966(CHEMBL406775)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376957BDBM50376957(CHEMBL261554)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376943BDBM50376943(CHEMBL260878)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376960BDBM50376960(CHEMBL261525)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322844BDBM50322844(3-ethyl-1-propyl-8-(1H-pyrazol-4-yl)-1H-purine-2,6...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376950BDBM50376950(CHEMBL259130)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376936BDBM50376936(CHEMBL408266)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376948BDBM50376948(CHEMBL259300)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376963BDBM50376963(CHEMBL430050)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]CPX from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376949BDBM50376949(CHEMBL259524)
Affinity DataKi:  91nMAssay Description:Displacement of [125I]ABMECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376936BDBM50376936(CHEMBL408266)
Affinity DataKi:  92nMAssay Description:Displacement of [125I]ABMECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376953BDBM50376953(CHEMBL260976)
Affinity DataKi:  95nMAssay Description:Displacement of [125I]ABMECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376950BDBM50376950(CHEMBL259130)
Affinity DataKi:  107nMAssay Description:Displacement of [125I]ABMECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376956BDBM50376956(CHEMBL264952)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Cv Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50376969BDBM50376969(CHEMBL258686)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
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