Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 3222
LigandChemical structure of BindingDB Monomer ID 29546BDBM29546(benzimidazolone scaffold, 15d)
Affinity DataKi:  3.40nM ΔG°:  -50.3kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29549BDBM29549(benzimidazolone scaffold, 15g)
Affinity DataKi:  6nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29548BDBM29548(benzimidazolone scaffold, 15f)
Affinity DataKi:  6nM ΔG°:  -48.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29554BDBM29554(benzimidazolone scaffold, 15m)
Affinity DataKi:  7nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29553BDBM29553(benzimidazolone scaffold, 15k)
Affinity DataKi:  11nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29552BDBM29552(benzimidazolone scaffold, 15j)
Affinity DataKi:  12nM ΔG°:  -47.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29551BDBM29551(benzimidazolone scaffold, 15i)
Affinity DataKi:  20nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29540BDBM29540(benzimidazolone scaffold, 8h)
Affinity DataKi:  22nM ΔG°:  -45.5kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29544BDBM29544(benzimidazolone scaffold, 15b)
Affinity DataKi:  25nM ΔG°:  -45.1kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29548BDBM29548(benzimidazolone scaffold, 15f)
Affinity DataKi:  26nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29541BDBM29541(benzimidazolone scaffold, 17d)
Affinity DataKi:  26nM ΔG°:  -45.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29545BDBM29545(benzimidazolone scaffold, 15c)
Affinity DataKi:  26nM ΔG°:  -45.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29550BDBM29550(benzimidazolone scaffold, 15h)
Affinity DataKi:  33nM ΔG°:  -44.4kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29542BDBM29542(benzimidazolone scaffold, 17f)
Affinity DataKi:  36nM ΔG°:  -44.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29550BDBM29550(benzimidazolone scaffold, 15h)
Affinity DataKi:  38nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29546BDBM29546(benzimidazolone scaffold, 15d)
Affinity DataKi:  40nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29551BDBM29551(benzimidazolone scaffold, 15i)
Affinity DataKi:  48nM ΔG°:  -43.5kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29547BDBM29547(benzimidazolone scaffold, 15e)
Affinity DataKi:  48nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29553BDBM29553(benzimidazolone scaffold, 15k)
Affinity DataKi:  66nM ΔG°:  -42.6kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29552BDBM29552(benzimidazolone scaffold, 15j)
Affinity DataKi:  78nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29547BDBM29547(benzimidazolone scaffold, 15e)
Affinity DataKi:  84nM ΔG°:  -42.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29541BDBM29541(benzimidazolone scaffold, 17d)
Affinity DataKi:  168nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29537BDBM29537(benzimidazolone scaffold, 8e)
Affinity DataKi:  168nM ΔG°:  -40.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29539BDBM29539(benzimidazolone scaffold, 8g)
Affinity DataKi:  182nM ΔG°:  -40.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29545BDBM29545(benzimidazolone scaffold, 15c)
Affinity DataKi:  243nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29542BDBM29542(benzimidazolone scaffold, 17f)
Affinity DataKi:  267nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29549BDBM29549(benzimidazolone scaffold, 15g)
Affinity DataKi:  269nM ΔG°:  -39.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29540BDBM29540(benzimidazolone scaffold, 8h)
Affinity DataKi:  296nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29536BDBM29536(benzimidazolone scaffold, 8d)
Affinity DataKi:  340nM ΔG°:  -38.4kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29538BDBM29538(benzimidazolone scaffold, 8f)
Affinity DataKi:  375nM ΔG°:  -38.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29543BDBM29543(benzimidazolone scaffold, 15a)
Affinity DataKi:  392nM ΔG°:  -38.0kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29554BDBM29554(benzimidazolone scaffold, 15m)
Affinity DataKi:  454nM ΔG°:  -37.7kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29533BDBM29533(benzimidazolone scaffold, 8a)
Affinity DataKi:  467nM ΔG°:  -37.6kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29536BDBM29536(benzimidazolone scaffold, 8d)
Affinity DataKi:  566nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29534BDBM29534(benzimidazolone scaffold, 8b)
Affinity DataKi:  636nM ΔG°:  -36.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29535BDBM29535(benzimidazolone scaffold, 8c)
Affinity DataKi:  646nM ΔG°:  -36.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29535BDBM29535(benzimidazolone scaffold, 8c)
Affinity DataKi:  864nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29534BDBM29534(benzimidazolone scaffold, 8b)
Affinity DataKi:  902nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29543BDBM29543(benzimidazolone scaffold, 15a)
Affinity DataKi:  1.03E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29533BDBM29533(benzimidazolone scaffold, 8a)
Affinity DataKi:  1.23E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29544BDBM29544(benzimidazolone scaffold, 15b)
Affinity DataKi:  1.84E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29537BDBM29537(benzimidazolone scaffold, 8e)
Affinity DataKi:  1.87E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29539BDBM29539(benzimidazolone scaffold, 8g)
Affinity DataKi:  2.50E+3nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29538BDBM29538(benzimidazolone scaffold, 8f)
Affinity DataKi:  1.80E+4nMAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed