Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50004206
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataKi:  38nMAssay Description:Inhibition of HIV1 protease by Lineweaver-Burke methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataKi:  38nMAssay Description:Inhibition of HIV1 protease by Hanes methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 41nMAssay Description:Inhibition of HIV1 protease by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataKi:  50nMAssay Description:Inhibition of HIV1 protease by Dixon methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480048(CHEMBL466684)
Affinity DataKi:  2.62E+4nMAssay Description:Inhibition of HIV1 protease by Lineweaver-Burke methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480048(CHEMBL466684)
Affinity DataKi:  2.62E+4nMAssay Description:Inhibition of HIV1 protease by Hanes methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480043(CHEMBL466688)
Affinity DataKi:  3.43E+4nMAssay Description:Inhibition of HIV1 protease by Lineweaver-Burke methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480043(CHEMBL466688)
Affinity DataKi:  3.43E+4nMAssay Description:Inhibition of HIV1 protease by Hanes methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480048(CHEMBL466684)
Affinity DataKi:  3.48E+4nMAssay Description:Inhibition of HIV1 protease by Dixon methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480048(CHEMBL466684)
Affinity DataIC50: 3.72E+4nMAssay Description:Inhibition of HIV1 protease by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480043(CHEMBL466688)
Affinity DataKi:  4.39E+4nMAssay Description:Inhibition of HIV1 protease by Dixon methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480043(CHEMBL466688)
Affinity DataIC50: 4.45E+4nMAssay Description:Inhibition of HIV1 protease by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480047(CHEMBL466502)
Affinity DataKi:  9.60E+4nMAssay Description:Inhibition of HIV1 protease by Dixon methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480047(CHEMBL466502)
Affinity DataKi:  9.60E+4nMAssay Description:Inhibition of HIV1 protease by Hanes methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480047(CHEMBL466502)
Affinity DataKi:  9.90E+4nMAssay Description:Inhibition of HIV1 protease by Lineweaver-Burke methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480044(CHEMBL471433)
Affinity DataKi:  1.38E+5nMAssay Description:Inhibition of HIV1 protease by Dixon methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480044(CHEMBL471433)
Affinity DataKi:  1.49E+5nMAssay Description:Inhibition of HIV1 protease by Lineweaver-Burke methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480044(CHEMBL471433)
Affinity DataKi:  1.49E+5nMAssay Description:Inhibition of HIV1 protease by Hanes methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480044(CHEMBL471433)
Affinity DataIC50: 1.69E+5nMAssay Description:Inhibition of HIV1 protease by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480047(CHEMBL466502)
Affinity DataIC50: 2.04E+5nMAssay Description:Inhibition of HIV1 protease by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480049(CHEMBL512599)
Affinity DataKi:  2.86E+5nMAssay Description:Inhibition of HIV1 protease by Dixon methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480049(CHEMBL512599)
Affinity DataKi:  2.92E+5nMAssay Description:Inhibition of HIV1 protease by Hanes methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480049(CHEMBL512599)
Affinity DataKi:  2.92E+5nMAssay Description:Inhibition of HIV1 protease by Lineweaver-Burke methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480049(CHEMBL512599)
Affinity DataIC50: 3.41E+5nMAssay Description:Inhibition of HIV1 protease by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480042(CHEMBL466687)
Affinity DataKi:  4.54E+5nMAssay Description:Inhibition of HIV1 protease by Dixon methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480042(CHEMBL466687)
Affinity DataKi:  4.61E+5nMAssay Description:Inhibition of HIV1 protease by Hanes methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480042(CHEMBL466687)
Affinity DataKi:  4.61E+5nMAssay Description:Inhibition of HIV1 protease by Lineweaver-Burke methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480042(CHEMBL466687)
Affinity DataIC50: 5.43E+5nMAssay Description:Inhibition of HIV1 protease by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480046(CHEMBL511210)
Affinity DataIC50: 5.45E+5nMAssay Description:Inhibition of HIV1 protease by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480046(CHEMBL511210)
Affinity DataKi:  5.74E+5nMAssay Description:Inhibition of HIV1 protease by Lineweaver-Burke methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480046(CHEMBL511210)
Affinity DataKi:  5.77E+5nMAssay Description:Inhibition of HIV1 protease by Dixon methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480046(CHEMBL511210)
Affinity DataKi:  6.18E+5nMAssay Description:Inhibition of HIV1 protease by Hanes methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Lyon

Curated by ChEMBL
LigandPNGBDBM50480045(CHEMBL466085)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of HIV1 protease by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed