Affinity DataKi: 1.70nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 184nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 408nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human prostanoid DP receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human prostanoid TP receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human prostanoid TP receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human prostanoid DP receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.22E+3nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity to human CRTH2 receptor expressed in HEK293-EBNA cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 810nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK293-EBNA cells assessed as inhibition of forskolin-stimulated intracellular cAMP producti...More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair