Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50039500
TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379109BDBM50379109(CHEMBL2012678)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]R-PIA from rat forebrain adenosine receptor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379123BDBM50379123(CHEMBL2012679)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]R-PIA from rat forebrain adenosine receptor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379111BDBM50379111(CHEMBL2012674)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]R-PIA from rat forebrain adenosine receptor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379107BDBM50379107(CHEMBL2012686)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]R-PIA from rat forebrain adenosine receptor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379106BDBM50379106(CHEMBL2012684)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]R-PIA from rat forebrain adenosine receptor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379110BDBM50379110(CHEMBL2012675)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]R-PIA from rat forebrain adenosine receptor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379120BDBM50379120(CHEMBL2012682)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]R-PIA from rat forebrain adenosine receptor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379111BDBM50379111(CHEMBL2012674)
Affinity DataKi:  5.90nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379108BDBM50379108(CHEMBL2012687)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]R-PIA from rat forebrain adenosine receptor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379122BDBM50379122(CHEMBL2012680)
Affinity DataKi:  6.60nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379106BDBM50379106(CHEMBL2012684)
Affinity DataKi:  8.90nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21220BDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataEC50:  10.2nMAssay Description:Agonist activity at human recombinant adenosine receptor-1 expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379117BDBM50379117(CHEMBL2012688)
Affinity DataKi:  10.3nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379120BDBM50379120(CHEMBL2012682)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379126BDBM50379126(CHEMBL2012673)
Affinity DataKi:  12.1nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379116BDBM50379116(CHEMBL2012689)
Affinity DataKi:  15.2nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379114BDBM50379114(CHEMBL2012691)
Affinity DataKi:  16.5nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379121BDBM50379121(CHEMBL2012681)
Affinity DataKi:  32.4nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379112BDBM50379112(CHEMBL2012693)
Affinity DataKi:  40.4nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379107BDBM50379107(CHEMBL2012686)
Affinity DataEC50:  40.7nMAssay Description:Agonist activity at human recombinant adenosine receptor-1 expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379108BDBM50379108(CHEMBL2012687)
Affinity DataKi:  41.5nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379107BDBM50379107(CHEMBL2012686)
Affinity DataKi:  47.9nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379111BDBM50379111(CHEMBL2012674)
Affinity DataKi:  51.6nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379119BDBM50379119(CHEMBL2012683)
Affinity DataKi:  52nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379106BDBM50379106(CHEMBL2012684)
Affinity DataKi:  68.4nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379120BDBM50379120(CHEMBL2012682)
Affinity DataKi:  72.2nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379121BDBM50379121(CHEMBL2012681)
Affinity DataKi:  72.7nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379119BDBM50379119(CHEMBL2012683)
Affinity DataKi:  78.8nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379109BDBM50379109(CHEMBL2012678)
Affinity DataKi:  82.6nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379113BDBM50379113(CHEMBL2012692)
Affinity DataKi:  83.2nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379118BDBM50379118(CHEMBL2012685)
Affinity DataKi:  86.8nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379118BDBM50379118(CHEMBL2012685)
Affinity DataKi:  110nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379115BDBM50379115(CHEMBL2012690)
Affinity DataKi:  114nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379110BDBM50379110(CHEMBL2012675)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379127BDBM50379127(CHEMBL2012672)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379123BDBM50379123(CHEMBL2012679)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379126BDBM50379126(CHEMBL2012673)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379125BDBM50379125(CHEMBL2012676)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379123BDBM50379123(CHEMBL2012679)
Affinity DataKi:  236nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379109BDBM50379109(CHEMBL2012678)
Affinity DataKi:  315nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379127BDBM50379127(CHEMBL2012672)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379107BDBM50379107(CHEMBL2012686)
Affinity DataKi:  470nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379110BDBM50379110(CHEMBL2012675)
Affinity DataKi:  500nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379125BDBM50379125(CHEMBL2012676)
Affinity DataKi:  560nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379124BDBM50379124(CHEMBL2012677)
Affinity DataKi:  760nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379122BDBM50379122(CHEMBL2012680)
Affinity DataKi:  930nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379114BDBM50379114(CHEMBL2012691)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379124BDBM50379124(CHEMBL2012677)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379112BDBM50379112(CHEMBL2012693)
Affinity DataKi:  1.91E+3nMAssay Description:Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379109BDBM50379109(CHEMBL2012678)
Affinity DataKi:  2.45E+3nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine receptor-2A expressed in HEK293 cell membrane after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
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