Compile Data Set for Download or QSAR
Report error Found 83 Enz. Inhib. hit(s) with all data for entry = 50034228
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359261(CHEMBL1923617)
Affinity DataKi:  0.350nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359239(CHEMBL1923629)
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359250(CHEMBL1923640)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359252(CHEMBL1923642)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359259(CHEMBL1923610)
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359238(CHEMBL1923628)
Affinity DataKi:  4.80nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359238(CHEMBL1923628)
Affinity DataKi:  4.80nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359237(CHEMBL1923627)
Affinity DataKi:  5nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359233(CHEMBL1923623)
Affinity DataKi:  6.20nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359282(CHEMBL1923609)
Affinity DataKi:  6.40nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359236(CHEMBL1923626)
Affinity DataKi:  7nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359235(CHEMBL1923625)
Affinity DataKi:  7.30nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359237(CHEMBL1923627)
Affinity DataEC50:  8.20nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359247(CHEMBL1923637)
Affinity DataKi:  9nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359236(CHEMBL1923626)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359249(CHEMBL1923639)
Affinity DataKi:  12nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359262(CHEMBL1923621)
Affinity DataKi:  15nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359256(ULIMORELIN | CHEMBL1923502)
Affinity DataKi:  16nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359260(CHEMBL1923611)
Affinity DataKi:  16nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359262(CHEMBL1923621)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359251(CHEMBL1923641)
Affinity DataKi:  19nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359261(CHEMBL1923617)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359234(CHEMBL1923624)
Affinity DataKi:  21nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359259(CHEMBL1923610)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359281(CHEMBL1923608)
Affinity DataKi:  25nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359248(CHEMBL1923638)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359252(CHEMBL1923642)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359256(ULIMORELIN | CHEMBL1923502)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359269(CHEMBL1923620)
Affinity DataKi:  32nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359232(CHEMBL1923622)
Affinity DataKi:  34nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359267(CHEMBL1923618)
Affinity DataKi:  34nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359265(CHEMBL1923614)
Affinity DataKi:  35nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359258(CHEMBL1923512)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359260(CHEMBL1923611)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359283(CHEMBL1923616)
Affinity DataKi:  43nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359239(CHEMBL1923629)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359238(CHEMBL1923628)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359238(CHEMBL1923628)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359248(CHEMBL1923638)
Affinity DataKi:  56nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359253(CHEMBL1923643)
Affinity DataKi:  58nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359254(CHEMBL1923644)
Affinity DataKi:  61nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359257(CHEMBL1923504)
Affinity DataKi:  68nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359246(CHEMBL1923636)
Affinity DataKi:  78nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359245(CHEMBL1923635)
Affinity DataKi:  81nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359257(CHEMBL1923504)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359250(CHEMBL1923640)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359255(CHEMBL1923501)
Affinity DataKi:  86nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359268(CHEMBL1923619)
Affinity DataKi:  104nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359258(CHEMBL1923512)
Affinity DataKi:  120nMAssay Description:Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAppetite-regulating hormone(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50359255(CHEMBL1923501)
Affinity DataEC50:  134nMAssay Description:Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
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