Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50005663
TargetDelta-type opioid receptor(Rat)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50001465(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]-deltorphin 2 from delta opioid receptor in rat GH3 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50493436(CHEMBL2429963)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]-deltorphin 2 from delta opioid receptor in rat GH3 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50493435(CHEMBL2432066)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]-deltorphin 2 from delta opioid receptor in rat GH3 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50493436(CHEMBL2429963)
Affinity DataEC50:  830nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50493437(CHEMBL2432064)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-deltorphin 2 from delta opioid receptor in rat GH3 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50493438(CHEMBL2432065)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-deltorphin 2 from delta opioid receptor in rat GH3 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50493435(CHEMBL2432066)
Affinity DataEC50: >1.50E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50493437(CHEMBL2432064)
Affinity DataEC50: >1.50E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50493438(CHEMBL2432065)
Affinity DataEC50: >1.50E+3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed