Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50005958
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Non-competitive inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate after 1 hr by double-recipro...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Non-competitive inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate after 1 hr by double-recipro...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Non-competitive inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate after 1 hr by double-recipro...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataKi: 3.80E+4nMAssay Description:Competitive inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate after 1 hr by double-reciprocal ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HIV-1 GST-tagged integrase-His6-tagged LEDGF complex expressed in Escherichia coli BL21(DE3) using [32P]-labeled U5B/U5A DNA as substra...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of HIV-1 GST-tagged integrase-His6-tagged LEDGF complex expressed in Escherichia coli BL21(DE3) using [32P]-labeled U5B/U5A DNA as substra...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of HIV-1 GST-tagged integrase-His6-tagged LEDGF complex expressed in Escherichia coli BL21(DE3) using [32P]-labeled U5B/U5A DNA as substra...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 integrase G140S mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pr...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 GST-tagged integrase-His6-tagged LEDGF complex expressed in Escherichia coli BL21(DE3) using [32P]-labeled U5B/U5A DNA as substra...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 integrase N155H mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pr...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 integrase E138K mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pr...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 integrase E92Q mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pro...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of HIV-1 GST-tagged integrase-His6-tagged LEDGF complex expressed in Escherichia coli BL21(DE3) using [32P]-labeled U5B/U5A DNA as substra...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of HIV-1 integrase E138K mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pr...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-processing reac...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of HIV-1 integrase G140S mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pr...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of HIV-1 integrase N155H mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pr...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of HIV-1 integrase E92Q mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pro...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of HIV-1 integrase expressed in Escherichia coli using [32P]-labeled U5B-2/U5A DNA as substrate assessed as inhibition of strand transfer ...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mg2+More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mg2+More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 1.30E+5nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mg2+More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mg2+More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of HIV-1 GST-tagged integrase-His6-tagged LEDGF complex expressed in Escherichia coli BL21(DE3) using [32P]-labeled U5B/U5A DNA as substra...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of HIV-1 GST-tagged integrase-His6-tagged LEDGF complex expressed in Escherichia coli BL21(DE3) using [32P]-labeled U5B/U5A DNA as substra...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of HIV-1 GST-tagged integrase-His6-tagged LEDGF complex expressed in Escherichia coli BL21(DE3) using [32P]-labeled U5B/U5A DNA as substra...More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: >2.56E+5nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mg2+More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mn2+More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mn2+More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mn2+More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mn2+More data for this Ligand-Target Pair
TargetIntegrase(Human immunodeficiency virus type 1)
Lomonosov Moscow State University
Curated by ChEMBL
Lomonosov Moscow State University
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Displacement of [32P]-labeled U5B/U5A DNA from HIV-1 integrase expressed in Escherichia coli in presence of Mn2+More data for this Ligand-Target Pair
