Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50006058
TargetPresenilin-1(Human)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50496623BDBM50496623(CHEMBL3134498)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of gamma-secretase (unknown origin) using Notch1 substrate assessed as Notch1-NICD productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50496623BDBM50496623(CHEMBL3134498)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of gamma-secretase (unknown origin) using APP substrate assessed as amyloid-beta40 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50496624BDBM50496624(CHEMBL3134497)
Affinity DataIC50: 0.910nMAssay Description:Inhibition of gamma-secretase (unknown origin) using APP substrate assessed as amyloid-beta40 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50496624BDBM50496624(CHEMBL3134497)
Affinity DataIC50: 1nMAssay Description:Inhibition of gamma-secretase (unknown origin) using Notch1 substrate assessed as Notch1-NICD productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed