Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50045148
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataEC50:  2.49E+4nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046953(Pectolinarin)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM23208((1R,2R,5S,8R,9R,10R,13R,14R,17S,19R)-17-hydroxy-1,...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046954(CHEMBL3314492)
Affinity DataEC50:  900nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046955(CHEMBL3314493)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046956(CHEMBL3314494)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046957(CHEBI:66441 | SCOPARIC ACID A)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046958(4-EPI-SCOPADULCIC ACID B)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046959(CHEMBL3314495)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM23411(5,6,7-trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-...)
Affinity DataEC50:  1.64E+4nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50049395(5,7,4'-Trihydroxy-6-methoxyflavone | 5,7-Dihydroxy...)
Affinity DataEC50:  7.30E+3nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046962(CVD-0019903 | Hispidulin-7-Glucoside | Hispidulosi...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046970(CHEMBL3314496)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Institute of Chinese Materia Medica

Curated by ChEMBL
LigandPNGBDBM50046951(CHEBI:2382 | CHEMBL3314497)
Affinity DataEC50:  4.30E+3nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed