Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50006399
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 35804BDBM35804(3-(4-{2-[6-Amino-9-((2R,3R,4S,5S)-5-ethylcarbamoyl...)
Affinity DataKi:  503nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499695BDBM50499695(CHEMBL3740969)
Affinity DataKi:  3.50E+4nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499688BDBM50499688(CHEMBL3741465)
Affinity DataKi:  4.40E+4nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499696BDBM50499696(CHEMBL3741290)
Affinity DataKi:  6.40E+4nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499690BDBM50499690(CHEMBL3740152)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499689BDBM50499689(CHEMBL3741118)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499692BDBM50499692(CHEMBL3740409)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499691BDBM50499691(CHEMBL3740229)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499700BDBM50499700(CHEMBL3740044)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499697BDBM50499697(CHEMBL3742187)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499699BDBM50499699(CHEMBL3740794)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499698BDBM50499698(CHEMBL3741961)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499694BDBM50499694(CHEMBL3739476)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50499693BDBM50499693(CHEMBL3741891)
Affinity DataKi: >2.00E+5nMAssay Description:Displacement of [3H]-ZM24135 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed