Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50048208
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50174269BDBM50174269(1-Benzenesulfonyl-4-piperazin-1-yl-1H-indole | 1-(...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208218BDBM50208218(CHEMBL3883432)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human recombinant AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208263BDBM50208263(CHEMBL3884227)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8961BDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 2nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208217BDBM50208217(CHEMBL3884195)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208258BDBM50208258(CHEMBL3885186)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208254BDBM50208254(CHEMBL3883921)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8960BDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208256BDBM50208256(CHEMBL3884618)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208216BDBM50208216(CHEMBL3884690)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human recombinant AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208218BDBM50208218(CHEMBL3883432)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman's met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208260BDBM50208260(CHEMBL3884988)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman's met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208259BDBM50208259(CHEMBL3884704)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208262BDBM50208262(CHEMBL3884312)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208214BDBM50208214(CHEMBL3884858)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208258BDBM50208258(CHEMBL3885186)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208256BDBM50208256(CHEMBL3884618)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human recombinant AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208216BDBM50208216(CHEMBL3884690)
Affinity DataIC50: 10nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208253BDBM50208253(CHEMBL3884867)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208257BDBM50208257(CHEMBL3884709)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8960BDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 10nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman's met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208260BDBM50208260(CHEMBL3884988)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208261BDBM50208261(CHEMBL3885452)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208256BDBM50208256(CHEMBL3884618)
Affinity DataIC50: 12nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman's met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208218BDBM50208218(CHEMBL3883432)
Affinity DataIC50: 12nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208255BDBM50208255(CHEMBL3885238)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208258BDBM50208258(CHEMBL3885186)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208256BDBM50208256(CHEMBL3884618)
Affinity DataIC50: 14nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208216BDBM50208216(CHEMBL3884690)
Affinity DataIC50: 15nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman's met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208212BDBM50208212(CHEMBL3883443)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208213BDBM50208213(CHEMBL3884254)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208252BDBM50208252(CHEMBL3884154)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208260BDBM50208260(CHEMBL3884988)
Affinity DataIC50: 17nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208214BDBM50208214(CHEMBL3884858)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208214BDBM50208214(CHEMBL3884858)
Affinity DataIC50: 21nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8961BDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 24nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman's met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208258BDBM50208258(CHEMBL3885186)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208218BDBM50208218(CHEMBL3883432)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208216BDBM50208216(CHEMBL3884690)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208215BDBM50208215(CHEMBL3883620)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208260BDBM50208260(CHEMBL3884988)
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208258BDBM50208258(CHEMBL3885186)
Affinity DataIC50: 46nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman's met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208214BDBM50208214(CHEMBL3884858)
Affinity DataIC50: 57nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman's met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8961BDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 131nMAssay Description:Inhibition of human recombinant AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman'...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208252BDBM50208252(CHEMBL3884154)
Affinity DataIC50: 608nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208261BDBM50208261(CHEMBL3885452)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208259BDBM50208259(CHEMBL3884704)
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8960BDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208212BDBM50208212(CHEMBL3883443)
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208213BDBM50208213(CHEMBL3884254)
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2018
Entry Details Article
PubMed
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