Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50047924
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197353BDBM50197353(CHEMBL3932329)
Affinity DataIC50: 121nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197347BDBM50197347(Ebselen Diselenide)
Affinity DataIC50: 230nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197302BDBM50197302(CHEMBL3920474)
Affinity DataIC50: 320nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197323BDBM50197323(CHEMBL3931605)
Affinity DataIC50: 920nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197348BDBM50197348(CHEMBL3940631)
Affinity DataIC50: 935nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197313BDBM50197313(CHEMBL3930560)
Affinity DataIC50: 1.35E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197299BDBM50197299(CHEMBL3913676)
Affinity DataIC50: 2.07E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197303BDBM50197303(CHEMBL3892953)
Affinity DataIC50: 2.35E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34233BDBM34233(EBSELEN | 2-Phenyl-benzo[d]isoselenazol-3-one(Ebse...)
Affinity DataIC50: 2.43E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197304BDBM50197304(CHEMBL3913688)
Affinity DataIC50: 2.67E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197352BDBM50197352(CHEMBL3912588)
Affinity DataIC50: 3.43E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197344BDBM50197344(CHEMBL3903564)
Affinity DataIC50: 4.47E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 106944BDBM106944(US8592468, EbSe2)
Affinity DataIC50: 4.97E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197297BDBM50197297(CHEMBL3928799 | ebselen derivative 2d)
Affinity DataIC50: 5.44E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197342BDBM50197342(CHEMBL3912637)
Affinity DataIC50: 6.27E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197300BDBM50197300(CHEMBL3912164 | ebselen derivative 2e)
Affinity DataIC50: 6.79E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197346BDBM50197346(CHEMBL3919905)
Affinity DataIC50: 7.57E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197298BDBM50197298(CHEMBL3947694)
Affinity DataIC50: 8.85E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197343BDBM50197343(CHEMBL3940582)
Affinity DataIC50: 9.13E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197349BDBM50197349(CHEMBL3983492 | ebselen derivative 1e)
Affinity DataIC50: 9.98E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197301BDBM50197301(CHEMBL3922662 | ebselen derivative 1d)
Affinity DataIC50: 1.02E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 106945BDBM106945(US8592468, EbSe3)
Affinity DataIC50: 1.04E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197350BDBM50197350(CHEMBL3964347)
Affinity DataIC50: 1.09E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197351BDBM50197351(CHEMBL3894620)
Affinity DataIC50: 1.39E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197296BDBM50197296(CHEMBL3894673)
Affinity DataIC50: 2.43E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50197345BDBM50197345(CHEMBL3931557)
Affinity DataIC50: 1.19E+5nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed