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Found 13 Enz. Inhib. hit(s) with all data for entry = 50035754
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50367744(CHEMBL603175)
Affinity DataEC50:  3.00E+4nMAssay Description:Inhibition of [3H]-MCC binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50013075(2-(Indan-5-ylamino)-1,9-dihydro-purin-6-one | CHEM...)
Affinity DataEC50:  1.50E+4nMAssay Description:Inhibition of [3H]-MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50013074(2-(4-Butyl-phenylamino)-1,9-dihydro-purin-6-one | ...)
Affinity DataEC50:  5.00E+4nMAssay Description:Inhibition of [3H]-MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50013093(2-(3-Ethyl-4-methyl-phenylamino)-1,9-dihydro-purin...)
Affinity DataEC50:  7.00E+3nMAssay Description:Inhibition of (-)-[3H]-nicotine binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50013094(2-Phenylamino-1,9-dihydro-purin-6-one | 2-Phenylam...)
Affinity DataEC50:  8.00E+3nMAssay Description:Inhibition of [3H]-MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50123607(CHEMBL3143943)
Affinity DataEC50:  3.00E+3nMAssay Description:inhibition of (-)-[3H]-nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50405722(CHEMBL2092762)
Affinity DataEC50:  7.50E+4nMAssay Description:Inhibitory activity against Herpes simplex virus type-I specific thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50018915(2-(4-Butyl-phenylamino)-9-(2-hydroxy-ethoxymethyl)...)
Affinity DataEC50:  1.40E+5nMAssay Description:Inhibition of [3H]-MCC binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50123605(CHEMBL3143935)
Affinity DataEC50:  300nMAssay Description:Inhibition of [3H]-MCC binding to rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50405103(CHEMBL2115349)
Affinity DataEC50:  2.50E+4nMAssay Description:Inhibitory activity against Herpes simplex virus type-I specific thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50013095(2-p-Tolylamino-1,9-dihydro-purin-6-one | CHEMBL368...)
Affinity DataEC50:  5.00E+4nMAssay Description:Inhibitory activity against Herpes simplex virus type-I specific thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50013099(2-(3-Ethyl-phenylamino)-1,9-dihydro-purin-6-one | ...)
Affinity DataEC50:  3.00E+3nMAssay Description:Inhibitory activity against Herpes simplex virus type-I specific thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1 (strain SC16) (HHV-1) (Human h...)
Istituto Di Genetica Biochimica Ed Evoluzionistica

Curated by ChEMBL
LigandPNGBDBM50123606(CHEMBL3143941)
Affinity DataEC50:  4.00E+5nMAssay Description:inhibition of (-)-[3H]-nicotine binding to torpedo electroplax membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed