Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50003046
TargetCalpain-1 catalytic subunit(Pig)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50363928(CHEMBL1951575)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50466172(CHEMBL366254 | PD-150606)
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of porcine Calpain-1 active site domain using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50466172(CHEMBL366254 | PD-150606)
Affinity DataIC50: 1.93E+4nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50466175(CHEMBL4289886)
Affinity DataIC50: 2.05E+4nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50466174(CHEMBL4293475)
Affinity DataIC50: 2.97E+4nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50466173(CHEMBL4288775)
Affinity DataIC50: 4.11E+4nMAssay Description:Inhibition of porcine Calpain-1 active site domain using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50466173(CHEMBL4288775)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of full length porcine Calpain-1 complex using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50363928(CHEMBL1951575)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of porcine Calpain-1 active site domain using (H2NeK(-FAM)-EVYGMMK(DABCYL)eOH) substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed