Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50012082
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554009BDBM50554009(CHEMBL4787992)
Affinity DataIC50: 0.0501nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554014BDBM50554014(CHEMBL4751860)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554012BDBM50554012(CHEMBL4764067)
Affinity DataIC50: 0.219nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554013BDBM50554013(CHEMBL4786278)
Affinity DataIC50: 0.295nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554010BDBM50554010(CHEMBL4795982)
Affinity DataIC50: 0.302nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554011BDBM50554011(CHEMBL4750105)
Affinity DataIC50: 0.302nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554001BDBM50554001(CHEMBL4789383)
Affinity DataIC50: 0.550nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257231BDBM50257231(CHEMBL4065973)
Affinity DataIC50: 0.603nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554007BDBM50554007(CHEMBL4740668)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553994BDBM50553994(CHEMBL4753692)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553993BDBM50553993(CHEMBL4744011)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553999BDBM50553999(CHEMBL4759447)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553992BDBM50553992(CHEMBL4797426)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554008BDBM50554008(CHEMBL4758442)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553998BDBM50553998(CHEMBL4788623)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554003BDBM50554003(CHEMBL4755954)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554002BDBM50554002(CHEMBL4775988)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554009BDBM50554009(CHEMBL4787992)
Affinity DataEC50:  1.90nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554000BDBM50554000(CHEMBL4799454)
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553995BDBM50553995(CHEMBL4761000)
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553991BDBM50553991(CHEMBL4745212)
Affinity DataIC50: 2.20nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554007BDBM50554007(CHEMBL4740668)
Affinity DataEC50:  2.40nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553997BDBM50553997(CHEMBL4763310)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554010BDBM50554010(CHEMBL4795982)
Affinity DataEC50:  2.40nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554001BDBM50554001(CHEMBL4789383)
Affinity DataEC50:  2.5nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554006BDBM50554006(CHEMBL4744024)
Affinity DataIC50: 2.5nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554002BDBM50554002(CHEMBL4775988)
Affinity DataEC50:  2.90nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553996BDBM50553996(CHEMBL4794535)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554005BDBM50554005(CHEMBL4741692)
Affinity DataIC50: 3.30nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554008BDBM50554008(CHEMBL4758442)
Affinity DataEC50:  3.5nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257231BDBM50257231(CHEMBL4065973)
Affinity DataEC50:  4.90nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553997BDBM50553997(CHEMBL4763310)
Affinity DataEC50:  4.90nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553994BDBM50553994(CHEMBL4753692)
Affinity DataEC50:  5.40nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553993BDBM50553993(CHEMBL4744011)
Affinity DataEC50:  6.20nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554000BDBM50554000(CHEMBL4799454)
Affinity DataEC50:  6.20nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554004BDBM50554004(CHEMBL4760648)
Affinity DataIC50: 6.30nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554004BDBM50554004(CHEMBL4760648)
Affinity DataEC50:  7.80nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554003BDBM50554003(CHEMBL4755954)
Affinity DataEC50:  8.10nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554006BDBM50554006(CHEMBL4744024)
Affinity DataEC50:  17nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553998BDBM50553998(CHEMBL4788623)
Affinity DataEC50:  26nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553992BDBM50553992(CHEMBL4797426)
Affinity DataEC50:  40nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553996BDBM50553996(CHEMBL4794535)
Affinity DataEC50:  49nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554005BDBM50554005(CHEMBL4741692)
Affinity DataEC50:  54nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553991BDBM50553991(CHEMBL4745212)
Affinity DataEC50:  74nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553999BDBM50553999(CHEMBL4759447)
Affinity DataEC50:  89nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
University of Alberta

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553995BDBM50553995(CHEMBL4761000)
Affinity DataEC50: <200nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed