Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50015071
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397360BDBM50397360(CHEMBL2170177 | US10188756, Compound CN110)
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50207561BDBM50207561(N-hydroxy-2,2-diphenylacetamide | CHEMBL396097 | C...)
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582532BDBM50582532(CHEMBL5085545)
Affinity DataEC50:  245nMAssay Description:Partial agonist activity at Gal4-fused human PPARgamma LBD in HepG2 cells assessed as transactivation incubated for 20 hrs measured by luminometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582535BDBM50582535(CHEMBL5087514)
Affinity DataEC50:  359nMAssay Description:Partial agonist activity at Gal4-fused human PPARgamma LBD in HepG2 cells assessed as transactivation incubated for 20 hrs measured by luminometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582546BDBM50582546(CHEMBL5083726)
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582535BDBM50582535(CHEMBL5087514)
Affinity DataIC50: 550nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582538BDBM50582538(CHEMBL5091419)
Affinity DataEC50:  729nMAssay Description:Partial agonist activity at Gal4-fused human PPARgamma LBD in HepG2 cells assessed as transactivation incubated for 20 hrs measured by luminometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582541BDBM50582541(CHEMBL5084422)
Affinity DataEC50:  791nMAssay Description:Partial agonist activity at Gal4-fused human PPARgamma LBD in HepG2 cells assessed as transactivation incubated for 20 hrs measured by luminometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582542BDBM50582542(CHEMBL5094339)
Affinity DataIC50: 840nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582544BDBM50582544(CHEMBL5073547)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582532BDBM50582532(CHEMBL5085545)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582537BDBM50582537(CHEMBL5073824)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582547BDBM50582547(CHEMBL5082258)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582526BDBM50582526(CHEMBL5089555)
Affinity DataEC50:  1.22E+3nMAssay Description:Partial agonist activity at Gal4-fused human PPARgamma LBD in HepG2 cells assessed as transactivation incubated for 20 hrs measured by luminometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582525BDBM50582525(CHEMBL5072376)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582530BDBM50582530(CHEMBL5090794)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582540BDBM50582540(CHEMBL5085291)
Affinity DataEC50:  1.61E+3nMAssay Description:Partial agonist activity at Gal4-fused human PPARgamma LBD in HepG2 cells assessed as transactivation incubated for 20 hrs measured by luminometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582526BDBM50582526(CHEMBL5089555)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582543BDBM50582543(CHEMBL5092097)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582540BDBM50582540(CHEMBL5085291)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582541BDBM50582541(CHEMBL5084422)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582524BDBM50582524(CHEMBL5089186)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582550BDBM50582550(CHEMBL5085184)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582528BDBM50582528(CHEMBL5086747)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582546BDBM50582546(CHEMBL5083726)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582538BDBM50582538(CHEMBL5091419)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582548BDBM50582548(CHEMBL5078917)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582529BDBM50582529(CHEMBL5082106)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582534BDBM50582534(CHEMBL5093916)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582540BDBM50582540(CHEMBL5085291)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582539BDBM50582539(CHEMBL5081178)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582524BDBM50582524(CHEMBL5089186)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582527BDBM50582527(CHEMBL5082287)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582545BDBM50582545(CHEMBL5076630)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582533BDBM50582533(CHEMBL5091605)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582531BDBM50582531(CHEMBL5090922)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582547BDBM50582547(CHEMBL5082258)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582525BDBM50582525(CHEMBL5072376)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582542BDBM50582542(CHEMBL5094339)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582535BDBM50582535(CHEMBL5087514)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582537BDBM50582537(CHEMBL5073824)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582530BDBM50582530(CHEMBL5090794)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582526BDBM50582526(CHEMBL5089555)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582549BDBM50582549(CHEMBL5090204)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582549BDBM50582549(CHEMBL5090204)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50397360BDBM50397360(CHEMBL2170177 | US10188756, Compound CN110)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582550BDBM50582550(CHEMBL5085184)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582538BDBM50582538(CHEMBL5091419)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582548BDBM50582548(CHEMBL5078917)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of recombinant human HDAC8 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Bharati Vidyapeeth'S College of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50582536BDBM50582536(CHEMBL5082458)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys (trifluoroacetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
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