Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50014910
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241089BDBM50241089(CHEMBL415049 | AZD1152, 33 | 2-(ethyl(3-(4-(5-(2-(...)
Affinity DataIC50: 0.370nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31837BDBM31837(Aurora Inhibitor, 35 | 2,4-Bisanilinopyrimidine, 1...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50277545BDBM50277545(Alisertib | MLN8237 | CHEMBL483158 | 4-(9-chloro-7...)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581040BDBM50581040(CHEMBL5075431)
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581041BDBM50581041(CHEMBL5091638)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581045BDBM50581045(CHEMBL5089708)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581042BDBM50581042(CHEMBL5078946)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581043BDBM50581043(CHEMBL5074672)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581052BDBM50581052(CHEMBL5078321)
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581044BDBM50581044(CHEMBL5078175)
Affinity DataIC50: 41nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581046BDBM50581046(CHEMBL5083318)
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581051BDBM50581051(CHEMBL5083583)
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581047BDBM50581047(CHEMBL5089253)
Affinity DataIC50: 48nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581055BDBM50581055(CHEMBL5082734)
Affinity DataIC50: 51nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581049BDBM50581049(CHEMBL5079532)
Affinity DataIC50: 52nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581054BDBM50581054(CHEMBL5076754)
Affinity DataIC50: 57nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581050BDBM50581050(CHEMBL5070908)
Affinity DataIC50: 58nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581048BDBM50581048(CHEMBL5093246)
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581056BDBM50581056(CHEMBL5073036)
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581053BDBM50581053(CHEMBL5076227)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581057BDBM50581057(CHEMBL5076654)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581058BDBM50581058(CHEMBL5073191)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581059BDBM50581059(CHEMBL5086056)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Taiwan National Health Research Institutes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50581060BDBM50581060(CHEMBL5081003)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant GST-tagged N-terminal truncated human Aurora A (123 to 401 residues) expressed in Sf9 insect cell using tetra-LRRASLG pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed