Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50015229
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584214(CHEMBL5082399)
Affinity DataKd:  230nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant using N-alpha-(6-FAM)-N-epsilon-(4-Iodophenylbutanoyl)-D-lysine as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584207(CHEMBL5091083)
Affinity DataKd:  340nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584199(CHEMBL5093073)
Affinity DataKd:  360nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584198(CHEMBL5078842)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584204(CHEMBL5082631)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584198(CHEMBL5078842)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584200(CHEMBL5083438)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584193(CHEMBL5076110)
Affinity DataKd:  3.20E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584194(CHEMBL5089368)
Affinity DataKd:  3.20E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584203(CHEMBL5091156)
Affinity DataKd:  3.50E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584206(CHEMBL5088591)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584209(CHEMBL5094773)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584205(CHEMBL5072994)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584197(CHEMBL5093280)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584193(CHEMBL5076110)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584195(CHEMBL5093981)
Affinity DataKd:  7.30E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584193(CHEMBL5076110)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584208(CHEMBL5071902)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584196(CHEMBL5075340)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584194(CHEMBL5089368)
Affinity DataKd:  9.00E+3nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584202(CHEMBL5085479)
Affinity DataKd:  2.60E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584201(CHEMBL5091965)
Affinity DataKd:  3.60E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584210(CHEMBL5079936)
Affinity DataKd:  7.00E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50009859((RS)-ibuprofen | CHEMBL521 | 2-(4-isobutylphenyl)p...)
Affinity DataKd:  7.30E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584213(CHEMBL5078753)
Affinity DataKd:  8.00E+4nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584212(CHEMBL5074099)
Affinity DataKd:  1.00E+5nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM50584211(CHEMBL5093259)
Affinity DataKd:  1.10E+5nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by fluorescence based competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetAlbumin(Human)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataKd:  1.20E+5nMAssay Description:Binding affinity to human serum albumin assessed as dissociation constant and measured after 5 mins by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)