Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50018946
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614092(CHEMBL5287112)
Affinity DataKi:  1.15E+3nMAssay Description:Competitive inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614093(CHEMBL5273859)
Affinity DataKi:  3.42E+3nMAssay Description:Competitive inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614092(CHEMBL5287112)
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614090(CHEMBL5269242)
Affinity DataKi:  4.60E+3nMAssay Description:Competitive inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614090(CHEMBL5269242)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human 20S immuno proteosome beta5i subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614090(CHEMBL5269242)
Affinity DataIC50: 6.65E+3nMAssay Description:Inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614092(CHEMBL5287112)
Affinity DataIC50: 8.44E+3nMAssay Description:Inhibition of human 20S immuno proteosome beta5i subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614091(CHEMBL5286864)
Affinity DataKi:  9.69E+3nMAssay Description:Competitive inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614093(CHEMBL5273859)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614091(CHEMBL5286864)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614093(CHEMBL5273859)
Affinity DataIC50: 2.21E+4nMAssay Description:Inhibition of human 20S immuno proteosome beta5i subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614091(CHEMBL5286864)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of human 20S immuno proteosome beta5i subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614085(CHEMBL5267503)
Affinity DataIC50: 2.01E+5nMAssay Description:Inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614088(CHEMBL5291286)
Affinity DataIC50: 4.40E+5nMAssay Description:Inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614089(CHEMBL5277601)
Affinity DataIC50: 4.91E+5nMAssay Description:Inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614087(CHEMBL5287265)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Middlesex University

Curated by ChEMBL
LigandPNGBDBM50614086(CHEMBL5266432)
Affinity DataIC50: 5.60E+5nMAssay Description:Inhibition of human 20S constitutive proteosome beta5c subunit using Suc-LLVY-AMC as substrate measured after 10 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed