Compile Data Set for Download or QSAR
Report error Found 93 Enz. Inhib. hit(s) with all data for entry = 50022429
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at recombinant human RAR-beta expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652169(CHEMBL5639513)
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  7.20nMAssay Description:Agonist activity at recombinant human RAR-gamma expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50178961(CHEMBL2385268)
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50178961(CHEMBL2385268)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at recombinant human RAR-beta expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50178961(CHEMBL2385268)
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at recombinant human RAR-alpha expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50055112(4-[(5,5-Dimethyl-8-thiophen-2-yl-5,6-dihydro-napht...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at recombinant human RAR-beta expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652183(CHEMBL5647012)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652168(CHEMBL5640022)
Affinity DataEC50:  25nMAssay Description:Agonist activity at recombinant human RAR-beta expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50471287(CHEMBL81176)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50471287(CHEMBL81176)
Affinity DataEC50:  55nMAssay Description:Agonist activity at recombinant human RAR-beta expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652169(CHEMBL5639513)
Affinity DataEC50:  75nMAssay Description:Agonist activity at recombinant human RAR-beta expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50178961(CHEMBL2385268)
Affinity DataEC50:  120nMAssay Description:Agonist activity at recombinant human RAR-gamma expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652183(CHEMBL5647012)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652168(CHEMBL5640022)
Affinity DataIC50: 140nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652171(CHEMBL5646471)
Affinity DataIC50: 173nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50178961(CHEMBL2385268)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human RAR-gamma transfected in human HeLa cells co-transfected with RARE-CAT reporter gene assessed as inhibition of ATRA-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50178961(CHEMBL2385268)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human RAR-beta transfected in human HeLa cells co-transfected with RARE-CAT reporter gene assessed as inhibition of ATRA-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50178961(CHEMBL2385268)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human RAR-alpha transfected in human HeLa cells co-transfected with RARE-CAT reporter gene assessed as inhibition of ATRA-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM36811(BMS614)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM36811(BMS614)
Affinity DataIC50: 270nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652169(CHEMBL5639513)
Affinity DataIC50: 310nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652182(CHEMBL5646931)
Affinity DataIC50: 350nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50471289(CHEMBL310790)
Affinity DataIC50: 430nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50055112(4-[(5,5-Dimethyl-8-thiophen-2-yl-5,6-dihydro-napht...)
Affinity DataIC50: 440nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652169(CHEMBL5639513)
Affinity DataEC50:  520nMAssay Description:Agonist activity at recombinant human RAR-gamma expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652171(CHEMBL5646471)
Affinity DataIC50: 520nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652168(CHEMBL5640022)
Affinity DataEC50:  560nMAssay Description:Agonist activity at recombinant human RAR-gamma expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652177(CHEMBL5639386)
Affinity DataIC50: 730nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652174(CHEMBL5641574)
Affinity DataIC50: 840nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652170(CHEMBL5646569)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652170(CHEMBL5646569)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652178(CHEMBL5641562)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50471287(CHEMBL81176)
Affinity DataIC50: 2.60E+3nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM36811(BMS614)
Affinity DataIC50: 2.70E+3nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652186(CHEMBL5647040)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652185(CHEMBL5647354)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652184(CHEMBL5641823)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652188(CHEMBL5647594)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652187(CHEMBL5647148)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-gamma expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor gamma(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50471287(CHEMBL81176)
Affinity DataEC50: >3.30E+3nMAssay Description:Agonist activity at recombinant human RAR-gamma expressed in mammalian cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652172(CHEMBL5646902)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50471287(CHEMBL81176)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50178961(CHEMBL2385268)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652188(CHEMBL5647594)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor alpha(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652187(CHEMBL5647148)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-alpha expressed in mammalian cells in presence of 9-cis-RA by luciferase reporter gene based transactiva...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652170(CHEMBL5646569)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652168(CHEMBL5640022)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor beta(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50652173(CHEMBL5639172)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at recombinant human RAR-beta expressed in mammalian cells in presence of ATRA by luciferase reporter gene based transactivation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
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