Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50020033
TargetNicotinamide phosphoribosyltransferase(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50625739(CHEMBL5429026)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of recombinant human NAMPT preincubated for 5 mins followed by NAM addition measured for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM81395(APO-866 | US20240327418, Example FK866 | US2024030...)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of recombinant human NAMPT preincubated for 5 mins followed by NAM addition measured for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNicotinamide phosphoribosyltransferase(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50625738(CHEMBL5437893)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of recombinant human NAMPT preincubated for 5 mins followed by NAM addition measured for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50625740(CHEMBL5439032)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant human NAMPT preincubated for 5 mins followed by NAM addition measured for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50625735(CHEMBL5413966)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of recombinant human NAMPT preincubated for 5 mins followed by NAM addition measured for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50625736(CHEMBL5416477)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant human NAMPT preincubated for 5 mins followed by NAM addition measured for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50625737(CHEMBL5435058)
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant human NAMPT preincubated for 5 mins followed by NAM addition measured for 15 mins by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed