Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50021132
Affinity DataKd: 7nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 8nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKd: 37nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 43nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataKd: 63nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataKd: 63nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 73nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 86nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 89nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataIC50: 96nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataIC50: 117nMAssay Description:Inhibition of VHL (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 120nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataKd: 129nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataKd: 134nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 149nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataKd: 186nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataKd: 305nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataKd: 528nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 640nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataKd: 740nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataIC50: 890nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of VHL/Elongin B/Elogin C (unknown origin) using FAM-DEALA-Hyp-YIPD as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.04E+3nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Binding affinity to NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate assessed as dissociation constant ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataIC50: 2.29E+3nMAssay Description:Inhibition of VHL (unknown origin) (1 to 213 residues)/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) using (FAM)-labeled HIF-1alpha pept...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of VHL/Elongin B/Elogin C (unknown origin) using FAM-DEALA-Hyp-YIPD as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of VHL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataKd: 5.40E+3nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 6.24E+3nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of VHL (unknown origin) (1 to 213 residues)/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) using (FAM)-labeled HIF-1alpha pept...More data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of VHL/Elongin B/Elogin C (unknown origin) using FAM-DEALA-Hyp-YIPD as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo as substrate incubated for 1 hrs by tracer based Nano...More data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of VHL/Elongin B/Elogin C (unknown origin) using FAM-DEALA-Hyp-YIPD as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair



































3D Structure (crystal)