Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50021637
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50370232(BA-41166E | L-5103 | Rifadin | Rifampicin | RIFAMP...)
Affinity DataKd:  9.40nMAssay Description:Binding affinity to Mycobacterium tuberculosis DprE1 assessed as dissociation constant by biolayer interferometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50642927(CHEMBL5591178)
Affinity DataKd:  1.35E+3nMAssay Description:Binding affinity to Mycobacterium tuberculosis DprE1 assessed as dissociation constant by biolayer interferometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50515570(Macozinone | PBTZ-169 | PBTZ169)
Affinity DataKd:  1.68E+3nMAssay Description:Binding affinity to Mycobacterium tuberculosis DprE1 assessed as dissociation constant by biolayer interferometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDecaprenylphosphoryl-beta-D-ribose oxidase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50642926(CHEMBL5574579)
Affinity DataKd:  2.50E+4nMAssay Description:Binding affinity to Mycobacterium tuberculosis DprE1 assessed as dissociation constant by biolayer interferometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed