Compile Data Set for Download or QSAR
Report error Found 77 Enz. Inhib. hit(s) with all data for entry = 50021053
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  5nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  12nMAssay Description:Inhibition of human CA2 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  25nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 30nMAssay Description:Inhibition of hypoxia induced VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 30nMAssay Description:Inhibition of VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636321(CHEMBL5567975)
Affinity DataIC50: 32nMAssay Description:Inhibition of hypoxia induced VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636320(CHEMBL5523449)
Affinity DataIC50: 35nMAssay Description:Inhibition of hypoxia induced VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636317(CHEMBL5542165)
Affinity DataIC50: 69nMAssay Description:Inhibition of hypoxia induced VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636334(CHEMBL5558406)
Affinity DataIC50: 82nMAssay Description:Inhibition of VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 139nMAssay Description:Inhibition of hypoxia induced VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 139nMAssay Description:Inhibition of VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  250nMAssay Description:Inhibition of human CA1 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636331(CHEMBL5562045)
Affinity DataKi:  480nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636333(CHEMBL5563731)
Affinity DataKi:  600nMAssay Description:Inhibition of human CA1 preincubated for 10 mins by stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636331(CHEMBL5562045)
Affinity DataKi:  830nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636332(CHEMBL5517864)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human CA1 by stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636321(CHEMBL5567975)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636317(CHEMBL5542165)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636321(CHEMBL5567975)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636317(CHEMBL5542165)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636318(CHEMBL5559628)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636320(CHEMBL5523449)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636322(CHEMBL5542863)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636318(CHEMBL5559628)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636320(CHEMBL5523449)
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636322(CHEMBL5542863)
Affinity DataKi:  6.10E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636319(CHEMBL5562546)
Affinity DataKi:  6.50E+3nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636319(CHEMBL5562546)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636329(CHEMBL5561433)
Affinity DataKi:  6.90E+3nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636324(CHEMBL5568260)
Affinity DataKi:  6.90E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataKi:  8.10E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636326(CHEMBL5556495)
Affinity DataKi:  8.20E+3nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636323(CHEMBL5563945)
Affinity DataKi:  8.70E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636329(CHEMBL5561433)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636326(CHEMBL5556495)
Affinity DataKi:  9.10E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636324(CHEMBL5568260)
Affinity DataKi:  9.10E+3nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636327(CHEMBL5560339)
Affinity DataKi:  9.30E+3nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 1(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human CA1 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human CA2 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636328(CHEMBL5527931)
Affinity DataKi:  1.13E+4nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636327(CHEMBL5560339)
Affinity DataKi:  1.28E+4nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636328(CHEMBL5527931)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636330(CHEMBL5542880)
Affinity DataKi:  1.39E+4nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636325(CHEMBL5557106)
Affinity DataKi:  1.45E+4nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636325(CHEMBL5557106)
Affinity DataKi:  1.48E+4nMAssay Description:Inhibition of human CA2 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636330(CHEMBL5542880)
Affinity DataKi:  1.89E+4nMAssay Description:Inhibition of human CA9 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636323(CHEMBL5563945)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of human CA12 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636318(CHEMBL5559628)
Affinity DataKi:  6.34E+4nMAssay Description:Inhibition of human CA2 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarbonic anhydrase 2(Human)
Tanta University

Curated by ChEMBL
LigandPNGBDBM50636321(CHEMBL5567975)
Affinity DataKi:  7.43E+4nMAssay Description:Inhibition of human CA2 preincubated for 6 hrs by phenol red staining based stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
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