Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50021941
TargetE-selectin(Human)TBA
LigandPNGBDBM50646329(CHEMBL5590365)
Affinity DataKd:  740nMAssay Description:Binding affinity to E-selectin SCR2 domain (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646329(CHEMBL5590365)
Affinity DataKd:  910nMAssay Description:Binding affinity to sialyl LewisX mimetic 21a pretreated Blue-NHS-labelled E-selectin Lec-EGF/SCR1/SCR2 domain (unknown origin) measured after 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646328(CHEMBL5593230)
Affinity DataKd:  1.15E+3nMAssay Description:Binding affinity to sialyl LewisX mimetic 21a pretreated Blue-NHS-labelled E-selectin Lec-EGF/SCR1/SCR2 domain (unknown origin) measured after 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646330(CHEMBL5594959)
Affinity DataKd:  1.38E+3nMAssay Description:Binding affinity to sialyl LewisX mimetic 21a pretreated Blue-NHS-labelled E-selectin Lec-EGF/SCR1/SCR2 domain (unknown origin) measured after 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646327(CHEMBL5592583)
Affinity DataKd:  1.90E+3nMAssay Description:Binding affinity to E-selectin SCR2 domain (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646327(CHEMBL5592583)
Affinity DataKd:  1.90E+3nMAssay Description:Binding affinity to sialyl LewisX mimetic 21a pretreated Blue-NHS-labelled E-selectin Lec-EGF/SCR1/SCR2 domain (unknown origin) measured after 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646325(Rivipansel | GMI-1070 | PF-06460031)
Affinity DataKd:  4.30E+3nMAssay Description:Binding affinity to sialyl LewisX mimetic 21a pretreated Blue-NHS-labelled E-selectin Lec-EGF/SCR1/SCR2 domain (unknown origin) measured after 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646333(CHEMBL5595169)
Affinity DataKd:  8.40E+3nMAssay Description:Binding affinity to E-selectin SCR2 domain (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646332(CHEMBL5594888)
Affinity DataKd:  1.78E+4nMAssay Description:Binding affinity to E-selectin SCR2 domain (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646326(CHEMBL5592209)
Affinity DataKd:  2.63E+4nMAssay Description:Binding affinity to sialyl LewisX mimetic 21a pretreated Blue-NHS-labelled E-selectin Lec-EGF/SCR1/SCR2 domain (unknown origin) measured after 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646331(CHEMBL407747)
Affinity DataKd:  6.07E+4nMAssay Description:Binding affinity to E-selectin SCR2 domain (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetE-selectin(Human)TBA
LigandPNGBDBM50646324(CHEMBL5593432)
Affinity DataKd:  7.38E+5nMAssay Description:Binding affinity to sialyl LewisX mimetic 21a pretreated Blue-NHS-labelled E-selectin Lec-EGF/SCR1/SCR2 domain (unknown origin) measured after 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed