Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50022129
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648459BDBM50648459(CHEMBL5612801)
Affinity DataIC50: 5nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648458BDBM50648458(CHEMBL5612090)
Affinity DataIC50: 5nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648472BDBM50648472(CHEMBL5613571)
Affinity DataIC50: 5nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648452BDBM50648452(CHEMBL5613018)
Affinity DataIC50: 5nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648482BDBM50648482(CHEMBL5613568)
Affinity DataIC50: 5nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648464BDBM50648464(CHEMBL5614116)
Affinity DataIC50: 5nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648475BDBM50648475(CHEMBL5614294)
Affinity DataIC50: 8nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648480BDBM50648480(CHEMBL5613188)
Affinity DataIC50: 8nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648461BDBM50648461(CHEMBL5613166)
Affinity DataIC50: 9nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648483BDBM50648483(CHEMBL5613313)
Affinity DataIC50: 10nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647344BDBM50647344(CHEMBL5090908)
Affinity DataIC50: 11nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648449BDBM50648449(CHEMBL5612748)
Affinity DataIC50: 17nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648474BDBM50648474(CHEMBL5612433)
Affinity DataIC50: 18nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648484BDBM50648484(CHEMBL5613132)
Affinity DataIC50: 19nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648454BDBM50648454(CHEMBL5613734)
Affinity DataIC50: 23nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648473BDBM50648473(CHEMBL5612613)
Affinity DataIC50: 28nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648479BDBM50648479(CHEMBL5613913)
Affinity DataIC50: 29nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648462BDBM50648462(CHEMBL5613844)
Affinity DataIC50: 30nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648453BDBM50648453(CHEMBL5613375)
Affinity DataIC50: 30nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648465BDBM50648465(CHEMBL5614029)
Affinity DataIC50: 38nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648470BDBM50648470(CHEMBL5613660)
Affinity DataIC50: 40nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648478BDBM50648478(CHEMBL5612699)
Affinity DataIC50: 45nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648457BDBM50648457(CHEMBL5613840)
Affinity DataIC50: 51nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648455BDBM50648455(CHEMBL5613030)
Affinity DataIC50: 53nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648471BDBM50648471(CHEMBL5612884)
Affinity DataIC50: 58nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648466BDBM50648466(CHEMBL5612171)
Affinity DataIC50: 67nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648469BDBM50648469(CHEMBL5614261)
Affinity DataIC50: 83nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648481BDBM50648481(CHEMBL5612560)
Affinity DataIC50: 84nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648467BDBM50648467(CHEMBL5612286)
Affinity DataIC50: 86nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648450BDBM50648450(CHEMBL5612829)
Affinity DataIC50: 93nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648460BDBM50648460(CHEMBL5614357)
Affinity DataIC50: 111nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648451BDBM50648451(CHEMBL5611969)
Affinity DataIC50: 117nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648468BDBM50648468(CHEMBL5612643)
Affinity DataIC50: 221nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648476BDBM50648476(CHEMBL5613187)
Affinity DataIC50: 430nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648456BDBM50648456(CHEMBL5612551)
Affinity DataIC50: 712nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648477BDBM50648477(CHEMBL5611945)
Affinity DataIC50: 728nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50648463BDBM50648463(CHEMBL5614141)
Affinity DataIC50: 803nMAssay Description:Inverse agonist activity at Pseudomonas aeruginosa PqsR extracted from Escherichia coli Dh5alpha co-expressing lacZ incubated with test compound in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed