Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50005472
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035320(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  1.30nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035303((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  1.40nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037272((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  1.70nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035326(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  1.80nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035305((S)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  2nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035328((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  2.70nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035324((S)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  2.90nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035330(R-(+)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  7nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  8.70nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035329((+/-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  12nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035306((1-Chloro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  12.6nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035307(S-(-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  14nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50020222(CHEMBL285755 | 7-Dipropylamino-5,6,7,8-tetrahydro-...)
Affinity DataKi:  54nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035330(R-(+)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  100nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035320(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  120nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037274(Dipropyl-(6,7,8,9-tetrahydro-1H-benzo[g]indol-8-yl...)
Affinity DataKi:  145nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035307(S-(-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  146nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035329((+/-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  156nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035301(Dipropyl-[1-(2,2,2-trifluoro-ethyl)-6,7,8,9-tetrah...)
Affinity DataKi:  182nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037274(Dipropyl-(6,7,8,9-tetrahydro-1H-benzo[g]indol-8-yl...)
Affinity DataKi:  220nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035306((1-Chloro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  317nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037271(Dipropyl-(5,6,7,8-tetrahydro-1H-benzo[f]indol-7-yl...)
Affinity DataKi:  350nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035303((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  382nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037275((2,3,6,7,8,9-Hexahydro-1H-benzo[g]indol-8-yl)-dipr...)
Affinity DataKi:  410nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035328((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  419nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035326(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  439nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037272((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  538nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037276(8-Dipropylamino-2,3,6,7,8,9-hexahydro-benzo[g]indo...)
Affinity DataKi:  550nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037271(Dipropyl-(5,6,7,8-tetrahydro-1H-benzo[f]indol-7-yl...)
Affinity DataKi:  570nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037275((2,3,6,7,8,9-Hexahydro-1H-benzo[g]indol-8-yl)-dipr...)
Affinity DataKi:  650nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037277(7-Dipropylamino-5,6,7,8-tetrahydro-1H-benzo[f]indo...)
Affinity DataKi:  700nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035301(Dipropyl-[1-(2,2,2-trifluoro-ethyl)-6,7,8,9-tetrah...)
Affinity DataKi:  796nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037273(Dipropyl-[3-(2,2,2-trifluoro-ethyl)-6,7,8,9-tetrah...)
Affinity DataKi:  2.33E+3nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50020222(CHEMBL285755 | 7-Dipropylamino-5,6,7,8-tetrahydro-...)
Affinity DataKi:  2.81E+3nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035305((S)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  3.59E+3nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037277(7-Dipropylamino-5,6,7,8-tetrahydro-1H-benzo[f]indo...)
Affinity DataKi:  4.72E+3nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037278(8-Dipropylamino-6,7,8,9-tetrahydro-1H-benzo[g]indo...)
Affinity DataKi:  6.72E+3nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035324((S)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  8.02E+3nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037273(Dipropyl-[3-(2,2,2-trifluoro-ethyl)-6,7,8,9-tetrah...)
Affinity DataKi:  8.80E+3nMAssay Description:Displacement of the radioligand [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037276(8-Dipropylamino-2,3,6,7,8,9-hexahydro-benzo[g]indo...)
Affinity DataKi: >1.60E+4nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50037278(8-Dipropylamino-6,7,8,9-tetrahydro-1H-benzo[g]indo...)
Affinity DataKi: >1.60E+4nMAssay Description:Displacement of the radioligand [3H]spiperone from D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed