Compile Data Set for Download or QSAR
Report error Found 81 Enz. Inhib. hit(s) with all data for entry = 50006183
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045792BDBM50045792(3-[3,4-Dimethyl-1-(4-methyl-pent-4-enyl)-piperidin...)
Affinity DataKi:  0.170nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045742BDBM50045742(3-[3,4-Dimethyl-1-(3-thiophen-3-yl-propyl)-piperid...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045776BDBM50045776(CHEMBL982 | Revex | Nalmetrene | ORF-11676 | cid_5...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045780BDBM50045780(3-[1-(3-Cyclohexyl-3-hydroxy-propyl)-3,4-dimethyl-...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045779BDBM50045779(3-[3,4-Dimethyl-1-(4-methyl-pentyl)-piperidin-4-yl...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045781BDBM50045781(1-Cyclohexyl-3-[4-(3-hydroxy-phenyl)-3,4-dimethyl-...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045791BDBM50045791(3-[1-(3-Cyclopentyl-propyl)-3,4-dimethyl-piperidin...)
Affinity DataKi:  0.370nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045786BDBM50045786(3-[1-(3-Cyclopentyl-3-hydroxy-propyl)-3,4-dimethyl...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045775BDBM50045775(3-[1-(3-Cyclohexyl-3-hydroxy-propyl)-3,4-dimethyl-...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045785BDBM50045785(3-[1-(3-Cyclohexyl-propyl)-3,4-dimethyl-piperidin-...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045735BDBM50045735(3-[1-(3-Hydroxy-3-thiophen-2-yl-propyl)-3,4-dimeth...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60212BDBM60212(SMR000058767 | NALTREXONE HYDROCHLORIDE | MLS00006...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045733BDBM50045733(3-[3,4-Dimethyl-1-(3-thiophen-2-yl-propyl)-piperid...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045733BDBM50045733(3-[3,4-Dimethyl-1-(3-thiophen-2-yl-propyl)-piperid...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045770BDBM50045770(3-(1-Heptyl-3,4-dimethyl-piperidin-4-yl)-phenol | ...)
Affinity DataKi:  0.620nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045778BDBM50045778(3-[1-(2-Cyclohexyl-ethyl)-3,4-dimethyl-piperidin-4...)
Affinity DataKi:  0.650nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045758BDBM50045758(3-[3,4-Dimethyl-1-(3-phenyl-propyl)-piperidin-4-yl...)
Affinity DataKi:  0.690nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045784BDBM50045784((3R,4R)3-[3,4-Dimethyl-1-(5-methyl-hexyl)-piperidi...)
Affinity DataKi:  0.890nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045784BDBM50045784((3R,4R)3-[3,4-Dimethyl-1-(5-methyl-hexyl)-piperidi...)
Affinity DataKi:  0.890nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045749BDBM50045749(3-[1-(3-Hydroxy-3-phenyl-propyl)-3,4-dimethyl-pipe...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045782BDBM50045782(3-[1-(2-Cyclopent-2-enyl-ethyl)-3,4-dimethyl-piper...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045738BDBM50045738((3R,4R)3-(1-Hexyl-3,4-dimethyl-piperidin-4-yl)-phe...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045738BDBM50045738((3R,4R)3-(1-Hexyl-3,4-dimethyl-piperidin-4-yl)-phe...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045789BDBM50045789(3-[3,4-Dimethyl-1-(5-methyl-hexyl)-piperidin-4-yl]...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045777BDBM50045777(3-[1-(3-Cyclohexyl-3-hydroxy-propyl)-3,4-dimethyl-...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045743BDBM50045743(3-[3,4-Dimethyl-1-(3-thiophen-2-yl-propyl)-piperid...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045784BDBM50045784((3R,4R)3-[3,4-Dimethyl-1-(5-methyl-hexyl)-piperidi...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045784BDBM50045784((3R,4R)3-[3,4-Dimethyl-1-(5-methyl-hexyl)-piperidi...)
Affinity DataKi:  1.91nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045775BDBM50045775(3-[1-(3-Cyclohexyl-3-hydroxy-propyl)-3,4-dimethyl-...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045776BDBM50045776(CHEMBL982 | Revex | Nalmetrene | ORF-11676 | cid_5...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045794BDBM50045794(3-[1-(3-Cyclohexyl-3-hydroxy-propyl)-3,4-dimethyl-...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045778BDBM50045778(3-[1-(2-Cyclohexyl-ethyl)-3,4-dimethyl-piperidin-4...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045790BDBM50045790(3-[1-(2-Cyclopentyl-ethyl)-3,4-dimethyl-piperidin-...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045785BDBM50045785(3-[1-(3-Cyclohexyl-propyl)-3,4-dimethyl-piperidin-...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045795BDBM50045795((3R,4R)3-[1-(3-Cyclohexyl-3-hydroxy-propyl)-3,4-di...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045783BDBM50045783(3-[1-(3-Hydroxy-4-methyl-pentyl)-3,4-dimethyl-pipe...)
Affinity DataKi:  2.60nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045789BDBM50045789(3-[3,4-Dimethyl-1-(5-methyl-hexyl)-piperidin-4-yl]...)
Affinity DataKi:  3nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045791BDBM50045791(3-[1-(3-Cyclopentyl-propyl)-3,4-dimethyl-piperidin...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045776BDBM50045776(CHEMBL982 | Revex | Nalmetrene | ORF-11676 | cid_5...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity towards delta-opioid receptor by displacement of [3H]DADL in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045781BDBM50045781(1-Cyclohexyl-3-[4-(3-hydroxy-phenyl)-3,4-dimethyl-...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045744BDBM50045744(3-(3,4-Dimethyl-1-pentyl-piperidin-4-yl)-phenol | ...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045780BDBM50045780(3-[1-(3-Cyclohexyl-3-hydroxy-propyl)-3,4-dimethyl-...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045738BDBM50045738((3R,4R)3-(1-Hexyl-3,4-dimethyl-piperidin-4-yl)-phe...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045738BDBM50045738((3R,4R)3-(1-Hexyl-3,4-dimethyl-piperidin-4-yl)-phe...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045775BDBM50045775(3-[1-(3-Cyclohexyl-3-hydroxy-propyl)-3,4-dimethyl-...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity towards delta-opioid receptor by displacement of [3H]DADL in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045786BDBM50045786(3-[1-(3-Cyclopentyl-3-hydroxy-propyl)-3,4-dimethyl...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045788BDBM50045788((3S,4S)3-(1-Hexyl-3,4-dimethyl-piperidin-4-yl)-phe...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]Nal in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045788BDBM50045788((3S,4S)3-(1-Hexyl-3,4-dimethyl-piperidin-4-yl)-phe...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60212BDBM60212(SMR000058767 | NALTREXONE HYDROCHLORIDE | MLS00006...)
Affinity DataKi:  6nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045733BDBM50045733(3-[3,4-Dimethyl-1-(3-thiophen-2-yl-propyl)-piperid...)
Affinity DataKi:  6.10nMAssay Description:Binding affinity towards kappa opioid receptor by displacement of [3H]EKC in guinea pig cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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