Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50044433 Sort by
TargetGlucocorticoid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50016931(CHEBI:31677 | Hydrocortisone Succinate | NSC-7576 ...)
Affinity DataKd:  190nMAssay Description:Displacement of 1 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucocorticoid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM13775([3H]cortisol | (1S,2R,10S,11S,14R,15S,17S)-14,17-d...)
Affinity DataKd:  43nMAssay Description:Displacement of 1 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucocorticoid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50016932(CHEMBL3273976)
Affinity DataKd:  7nMAssay Description:Displacement of 2 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucocorticoid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50016933(CHEMBL3273977)
Affinity DataKd:  430nMAssay Description:Displacement of 2 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016934(CHEBI:82520 | ESTRADIOL MUSTARD)
Affinity DataKd:  3.00E+3nMAssay Description:Displacement of radiolabeled estradiol from estradiol receptor in rat uterine cytosolMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed