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Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50044433
TargetGlucocorticoid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50016931(CHEBI:31677 | HYDROCORTISONE HEMISUCCINATE | Hydro...)
Affinity DataKd:  190nMAssay Description:Displacement of 1 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM13775((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...)
Affinity DataKd:  43nMAssay Description:Displacement of 1 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetEstrogen receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016934(CHEBI:82520 | ESTRADIOL MUSTARD)
Affinity DataKd:  3.00E+3nMAssay Description:Displacement of radiolabeled estradiol from estradiol receptor in rat uterine cytosolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50016933(CHEMBL3273977)
Affinity DataKd:  430nMAssay Description:Displacement of 2 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGlucocorticoid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50016932(CHEMBL3273976)
Affinity DataKd:  7nMAssay Description:Displacement of 2 x 10'-8 M of [1,2,3-3H]-triamcinolone acetonide from glucocorticoid receptor in soluble fraction of mouse L929 cells after 20 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed