Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50007264
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50454655(CHEMBL2111779)
Affinity DataKi:  6.10nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]GR-125743 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060519(3-(3-Dimethylamino-propyl)-4-hydroxy-N-(4-pyridin-...)
Affinity DataKi:  12.1nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060516(3-((E)-3-Dimethylamino-propenyl)-4-methoxy-N-(4-py...)
Affinity DataKi:  13.6nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060519(3-(3-Dimethylamino-propyl)-4-hydroxy-N-(4-pyridin-...)
Affinity DataKi:  14nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]GR-125743 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060518(3-(3-Dimethylamino-propyl)-4-methoxy-N-(4-pyridin-...)
Affinity DataKi:  15nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]GR-125743 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060517(3-(3-Dimethylamino-prop-1-ynyl)-4-methoxy-N-(4-pyr...)
Affinity DataKi:  16nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50454655(CHEMBL2111779)
Affinity DataKi:  19nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060516(3-((E)-3-Dimethylamino-propenyl)-4-methoxy-N-(4-py...)
Affinity DataKi:  19nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]GR-125743 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060517(3-(3-Dimethylamino-prop-1-ynyl)-4-methoxy-N-(4-pyr...)
Affinity DataKi:  22.3nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]GR-125743 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060518(3-(3-Dimethylamino-propyl)-4-methoxy-N-(4-pyridin-...)
Affinity DataKi:  70.1nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptor in C6-glial transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50454655(CHEMBL2111779)
Affinity DataKi:  169nMAssay Description:Binding affinity for 5-hydroxytryptamine 1D receptor in Cos-7 transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060518(3-(3-Dimethylamino-propyl)-4-methoxy-N-(4-pyridin-...)
Affinity DataKi:  540nMAssay Description:Binding affinity for 5-hydroxytryptamine 1D receptor in Cos-7 transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060516(3-((E)-3-Dimethylamino-propenyl)-4-methoxy-N-(4-py...)
Affinity DataKi:  560nMAssay Description:Binding affinity for 5-hydroxytryptamine 1D receptor in Cos-7 transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50454655(CHEMBL2111779)
Affinity DataKi:  633nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor in HeLa transfected cell type using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060519(3-(3-Dimethylamino-propyl)-4-hydroxy-N-(4-pyridin-...)
Affinity DataKi:  700nMAssay Description:Binding affinity for 5-hydroxytryptamine 1D receptor in Cos-7 transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060519(3-(3-Dimethylamino-propyl)-4-hydroxy-N-(4-pyridin-...)
Affinity DataKi:  842nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor in HeLa transfected cell type using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060518(3-(3-Dimethylamino-propyl)-4-methoxy-N-(4-pyridin-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor in HeLa transfected cell type using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060516(3-((E)-3-Dimethylamino-propenyl)-4-methoxy-N-(4-py...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor in HeLa transfected cell type using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060517(3-(3-Dimethylamino-prop-1-ynyl)-4-methoxy-N-(4-pyr...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor in HeLa transfected cell type using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50060517(3-(3-Dimethylamino-prop-1-ynyl)-4-methoxy-N-(4-pyr...)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 1D receptor in Cos-7 transfected cell type using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed