Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50007551
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408421(CHEMBL2113725)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)
Affinity DataIC50:  6nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408414(CHEMBL2113720)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408417(CHEMBL2113724)
Affinity DataIC50:  17nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408419(CHEMBL2113723)
Affinity DataIC50:  19nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408413(CHEMBL2113727)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408419(CHEMBL2113723)
Affinity DataIC50:  21nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408418(CHEMBL2113722)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408422(CHEMBL2113721)
Affinity DataIC50:  23nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408424(CHEMBL2113733)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50064506(1-Butyl-3-{3-methoxy-2-propoxy-5-[5-(3,4,5-trimeth...)
Affinity DataIC50:  33nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408422(CHEMBL2113721)
Affinity DataIC50:  33nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408423(CHEMBL2113726)
Affinity DataIC50:  38nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408415(CHEMBL2113730)
Affinity DataIC50:  39nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408418(CHEMBL2113722)
Affinity DataIC50:  43nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408417(CHEMBL2113724)
Affinity DataIC50:  45nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408413(CHEMBL2113727)
Affinity DataIC50:  58nMAssay Description:5-lipoxygenase inhibitory activity determined by measuring the conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cell using thin-layer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408415(CHEMBL2113730)
Affinity DataIC50:  71nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)
Affinity DataIC50:  94nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408414(CHEMBL2113720)
Affinity DataIC50:  100nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408421(CHEMBL2113725)
Affinity DataIC50:  118nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408424(CHEMBL2113733)
Affinity DataIC50:  161nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408420(CHEMBL2113731)
Affinity DataIC50:  167nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408416(CHEMBL2113732)
Affinity DataIC50:  285nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50029775((R)-(+)-N-{3-[5-(4-fluorophenoxy)furan-2-yl]-1-met...)
Affinity DataIC50:  298nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50064506(1-Butyl-3-{3-methoxy-2-propoxy-5-[5-(3,4,5-trimeth...)
Affinity DataIC50:  424nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408416(CHEMBL2113732)
Affinity DataIC50:  520nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50000541((+-)-1-(1-Benzo[b]thien-2-ylethyl)-1-hydroxyurea |...)
Affinity DataIC50:  804nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed