Compile Data Set for Download or QSAR
Report error Found 142 Enz. Inhib. hit(s) with all data for entry = 50041267
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408628BDBM50408628(CHEMBL139855)
Affinity DataIC50: 0.0126nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50114716BDBM50114716(N-[2-(2-Benzyl-5-methoxy-benzofuran-3-yl)-ethyl]-a...)
Affinity DataIC50: 0.0158nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50286970BDBM50286970(N-[2-(3H-Benzo[f]chromen-10-yl)-ethyl]-acetamide |...)
Affinity DataIC50: 0.158nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50286973BDBM50286973(N-[2-(2,3-Dihydro-1H-benzo[f]chromen-10-yl)-ethyl]...)
Affinity DataIC50: 0.251nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408640BDBM50408640(CHEMBL337764)
Affinity DataIC50: 0.316nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408584BDBM50408584(CHEMBL137998)
Affinity DataIC50: 0.794nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408657BDBM50408657(CHEMBL137878)
Affinity DataIC50: 0.794nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408555BDBM50408555(CHEMBL322762)
Affinity DataIC50: 0.794nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282765BDBM50282765(N-(6-Methoxy-9-methyl-2,3,4,9-tetrahydro-1H-carbaz...)
Affinity DataIC50: 1nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataIC50: 1nMAssay Description:Binding affinity for melatonin 1A receptor was measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408618BDBM50408618(CHEMBL138321)
Affinity DataIC50: 1nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 29611BDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataIC50: 1nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037253BDBM50037253(2-Iodo-N-[2-(5-methoxy-1H-indol-3-yl)-ethyl]-aceta...)
Affinity DataIC50: 1.26nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50286972BDBM50286972(N-(2-Naphtho[2,1-b]furan-9-yl-ethyl)-acetamide | C...)
Affinity DataIC50: 1.26nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408578BDBM50408578(CHEMBL417151)
Affinity DataIC50: 1.26nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037219BDBM50037219(N-[2-(5-Methoxy-benzo[b]thiophen-3-yl)-ethyl]-acet...)
Affinity DataIC50: 1.26nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037242BDBM50037242(N-[2-(5-Methoxy-benzofuran-3-yl)-ethyl]-acetamide ...)
Affinity DataIC50: 1.58nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408591BDBM50408591(CHEMBL138766)
Affinity DataIC50: 2nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037249BDBM50037249(Cyclopropanecarboxylic acid [2-(6-fluoro-5-methoxy...)
Affinity DataIC50: 2nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408556BDBM50408556(CHEMBL37771)
Affinity DataIC50: 2nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408631BDBM50408631(CHEMBL138817)
Affinity DataIC50: 2.51nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408649BDBM50408649(CHEMBL37703)
Affinity DataIC50: 2.51nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408600BDBM50408600(CHEMBL140549)
Affinity DataIC50: 3.16nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408551BDBM50408551(CHEMBL436006)
Affinity DataIC50: 3.16nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408579BDBM50408579(CHEMBL141115)
Affinity DataIC50: 3.16nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408560BDBM50408560(CHEMBL337580)
Affinity DataIC50: 3.98nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037222BDBM50037222(Cyclopropanecarboxylic acid [2-(5-methoxy-benzo[b]...)
Affinity DataIC50: 3.98nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408553BDBM50408553(CHEMBL335116)
Affinity DataIC50: 3.98nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408658BDBM50408658(CHEMBL441664)
Affinity DataIC50: 3.98nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037247BDBM50037247(Cyclopropanecarboxylic acid [2-(5-methoxy-benzofur...)
Affinity DataIC50: 5.01nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408601BDBM50408601(CHEMBL138440)
Affinity DataIC50: 5.01nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408559BDBM50408559(CHEMBL138752)
Affinity DataIC50: 5.01nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037228BDBM50037228(2-Iodo-N-[2-(5-methoxy-benzo[b]thiophen-3-yl)-ethy...)
Affinity DataIC50: 5.01nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408565BDBM50408565(CHEMBL137910)
Affinity DataIC50: 5.01nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408598BDBM50408598(CHEMBL139410)
Affinity DataIC50: 6.31nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037240BDBM50037240(Pentanoic acid [2-(5-methoxy-benzofuran-3-yl)-ethy...)
Affinity DataIC50: 6.31nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408563BDBM50408563(CHEMBL139014)
Affinity DataIC50: 6.31nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408625BDBM50408625(CHEMBL138549)
Affinity DataIC50: 7.94nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363763BDBM50363763(CHEMBL342432)
Affinity DataIC50: 7.94nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408614BDBM50408614(CHEMBL344268)
Affinity DataIC50: 7.94nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408604BDBM50408604(CHEMBL342655)
Affinity DataIC50: 7.94nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408648BDBM50408648(CHEMBL336010)
Affinity DataIC50: 7.94nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50286971BDBM50286971(N-[2-(2,3,7,8,9,10-Hexahydro-1H-benzo[f]chromen-10...)
Affinity DataIC50: 10nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408554BDBM50408554(CHEMBL341761)
Affinity DataIC50: 10nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408633BDBM50408633(CHEMBL138288)
Affinity DataIC50: 10nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408597BDBM50408597(CHEMBL344880)
Affinity DataIC50: 12.6nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408587BDBM50408587(CHEMBL342592)
Affinity DataIC50: 12.6nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408593BDBM50408593(CHEMBL336225)
Affinity DataIC50: 12.6nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408603BDBM50408603(CHEMBL139228)
Affinity DataIC50: 12.6nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Orleans University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408622BDBM50408622(CHEMBL139516)
Affinity DataIC50: 12.6nMAssay Description:Melatonin receptor type 1A binding affinity measured using 2-[125I]iodomelatonin on ovine pars tuberalis membrane homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
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