Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50007922
TargetProthrombin(Human)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294(1N-cyclopentyl-3-[4-amino(aminoimino)methylphenyl]...)
Affinity DataKi:  0.380nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294(1N-cyclopentyl-3-[4-amino(aminoimino)methylphenyl]...)
Affinity DataKi:  1.10nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069292(N-ethyl-N-cyclopentyl-3-(4-hydrazonoformamidepheny...)
Affinity DataKi:  4nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069293(N-methyl-N-n-butyl-3-(4-hydrazonoformamidephenyl)-...)
Affinity DataKi:  41nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069296(N-(n-propyl)-N-cyclopentyl-3-(4-hydrazonoformamide...)
Affinity DataKi:  93nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069298(N-methyl-N-cyclohexyl-3-(4-hydrazonoformamidepheny...)
Affinity DataKi:  152nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069299(N-(n-butyl)-N-cyclopentyl-3-(4-hydrazonoformamidep...)
Affinity DataKi:  231nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069295(N-methyl-N-cyclopropyl-3-(4-hydrazonoformamidephen...)
Affinity DataKi:  247nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069300(N-hydroxy-N-cyclopentyl-3-(4-hydrazonoformamidephe...)
Affinity DataKi:  367nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294(1N-cyclopentyl-3-[4-amino(aminoimino)methylphenyl]...)
Affinity DataKi:  1.10E+3nMAssay Description:The compound was tested for inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069297(1-[3-[4-amino(amineimino)methylphenyl]-2-(2-naphth...)
Affinity DataKi:  1.47E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Human)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294(1N-cyclopentyl-3-[4-amino(aminoimino)methylphenyl]...)
Affinity DataKi:  3.29E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Bovine)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069301(N-hydroxyethyl-N-cyclopentyl-3-(4-hydrazonoformami...)
Affinity DataKi:  7.04E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294(1N-cyclopentyl-3-[4-amino(aminoimino)methylphenyl]...)
Affinity DataKi:  2.72E+4nMAssay Description:The compound was tested for inhibitory activity against tissue plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294(1N-cyclopentyl-3-[4-amino(aminoimino)methylphenyl]...)
Affinity DataKi:  4.79E+4nMAssay Description:The compound was tested for inhibitory activity against human plasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed