Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50008250
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50065407((R)-N-((S)-1-Benzyl-2-oxo-ethyl)-3-benzyloxy-2-met...)
Affinity DataIC50: 11nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071828(Benzenesulfonic acid (3R,5S)-1-benzenesulfonyl-5-(...)
Affinity DataIC50: 13nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071825((R)-1-(Toluene-4-sulfonyl)-pyrrolidine-2-carboxyli...)
Affinity DataIC50: 14nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071823((2R,4R)-4-Azido-1-(toluene-4-sulfonyl)-pyrrolidine...)
Affinity DataIC50: 28nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071828(Benzenesulfonic acid (3R,5S)-1-benzenesulfonyl-5-(...)
Affinity DataIC50: 38nMAssay Description:Compound was tested for inhibitory activity against Cathepsin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071829((S)-1-Benzenesulfonyl-pyrrolidine-2-carboxylic aci...)
Affinity DataIC50: 41nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50065407((R)-N-((S)-1-Benzyl-2-oxo-ethyl)-3-benzyloxy-2-met...)
Affinity DataIC50: 42nMAssay Description:Compound was tested for inhibitory activity against Cathepsin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071827((S)-1-Methanesulfonyl-pyrrolidine-2-carboxylic aci...)
Affinity DataIC50: 45nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071826((R)-1-Methanesulfonyl-pyrrolidine-2-carboxylic aci...)
Affinity DataIC50: 53nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071824((2R,4R)-1-(Toluene-4-sulfonyl)-4-(2,2,2-trifluoro-...)
Affinity DataIC50: 100nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071830((2S,4R)-1-Benzenesulfonyl-4-benzyloxy-pyrrolidine-...)
Affinity DataIC50: 125nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071827((S)-1-Methanesulfonyl-pyrrolidine-2-carboxylic aci...)
Affinity DataIC50: 883nMAssay Description:Compound was tested for inhibitory activity against Cathepsin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071829((S)-1-Benzenesulfonyl-pyrrolidine-2-carboxylic aci...)
Affinity DataIC50: 1.40E+3nMAssay Description:Compound was tested for inhibitory activity against Cathepsin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071826((R)-1-Methanesulfonyl-pyrrolidine-2-carboxylic aci...)
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was tested for inhibitory activity against Cathepsin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071825((R)-1-(Toluene-4-sulfonyl)-pyrrolidine-2-carboxyli...)
Affinity DataIC50: 3.60E+3nMAssay Description:Compound was tested for inhibitory activity against Cathepsin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071822((2R,4R)-4-Cyano-1-(toluene-4-sulfonyl)-pyrrolidine...)
Affinity DataIC50: 8.70E+3nMAssay Description:Compound was tested for inhibitory activity against recombinant human Calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071822((2R,4R)-4-Cyano-1-(toluene-4-sulfonyl)-pyrrolidine...)
Affinity DataIC50: 8.70E+3nMAssay Description:Compound was tested for inhibitory activity against Cathepsin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50071823((2R,4R)-4-Azido-1-(toluene-4-sulfonyl)-pyrrolidine...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested for inhibitory activity against Cathepsin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed