Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50008368
TargetProtein kinase C alpha type(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50048888(Acetic acid 2-hydroxymethyl-5-oxo-4-tetradecyliden...)
Affinity DataKi:  35nMAssay Description:Displacement of [20-3H]-phorbol 12,13-dibutyrate (PDBU) from PKCalpha (C1b domain)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50048890(Acetic acid 2-hydroxymethyl-5-oxo-4-tetradec-(E)-y...)
Affinity DataKi:  78nMAssay Description:Displacement of [20-3H]-phorbol 12,13-dibutyrate (PDBU) from PKCalpha (C1b domain)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50072733(5-Ethoxymethyl-5-hydroxymethyl-3-tetradec-(E)-ylid...)
Affinity DataKi:  4.98E+3nMAssay Description:Displacement of [20-3H]-phorbol 12,13-dibutyrate (PDBU) from PKCalpha (C1b domain)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50072734(5-Ethoxymethyl-5-hydroxymethyl-3-tetradec-(Z)-ylid...)
Affinity DataKi:  7.46E+3nMAssay Description:Displacement of [20-3H]-phorbol 12,13-dibutyrate (PDBU) from PKCalpha (C1b domain)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Institutes of Health

Curated by ChEMBL
LigandPNGBDBM50072735(Acetic acid 2-hydroxymethyl-4-tetradec-(E)-ylidene...)
Affinity DataKi:  7.58E+3nMAssay Description:Displacement of [20-3H]-phorbol 12,13-dibutyrate (PDBU) from PKCalpha (C1b domain)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed