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Target
Bromodomain testis-specific protein [287-359]
Ligand
BDBM50103503
Substrate
n/a
Meas. Tech.
Plate-Based Time-Resolved Fluorescence Energy Transfer (TR-FRET) Assays
IC50
708±n/a nM
Citation
 Zhou, J; Brasier, AR; Tian, B; Liu, Z; Chen, H; Rytting, E Inhibitors of bromodomain-containing protein 4 (BRD4) US Patent  US11117865 Publication Date 9/14/2021 
Target
Name:
Bromodomain testis-specific protein [287-359]
Synonyms:
BRDT | BRDT_HUMAN | Bromodomain testis-specific protein (BRDT)(BD2)
Type:
n/a
Mol. Mass.:
8713.30
Organism:
Human
Description:
Q58F21[287-359]
Residue:
73
Sequence:
KHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVV
  
Inhibitor
Name:
BDBM50103503
Synonyms:
CHEMBL2393130 | US11117865, Compound RVX-208 | US20250221977, Compound RVX-208
Type:
Small organic molecule
Emp. Form.:
C20H22N2O5
Mol. Mass.:
370.15
SMILES:
Cc1cc(cc(c1OCCO)C)C2=Nc3cc(cc(c3C(=O)N2)OC)OC
Structure:
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