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Target
Bromodomain testis-specific protein [44-116]
Ligand
BDBM674567
Substrate
n/a
Meas. Tech.
AlphaScreen Assay
IC50
15.0±n/a nM
Citation
 Matzuk, M; Yu, Z; Ku, A; Anglin, J; Li, F; Young, D; Chen, Y; Ucisik, M; Faver, J; Palmer, S; Sharma, R; Kim, C BET SUBFAMILY INHIBITORS AND METHODS USING SAME US Patent  US20240158355 Publication Date 5/16/2024 
Target
Name:
Bromodomain testis-specific protein [44-116]
Synonyms:
Bromodomain testis-specific protein (BRDT)(BD1)(44-116)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
8758.44
Organism:
Homo sapiens (Human)
Description:
Sequence: Q58F21; Family & Domains; Bromo 1
Residue:
73
Sequence:
WKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIV
  
Inhibitor
Name:
BDBM674567
Synonyms:
US20240158355, Compound 7
Type:
Small organic molecule
Emp. Form.:
n/a
Mol. Mass.:
n/a
SMILES:
CNC(=O)c1ccc(cc1)C(=O)Nc1cc(NC(=O)c2ccc3n(C)nc(-c4ccc(N)cc4)c3c2)ccc1OC
Structure:
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