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Target
Bromodomain testis-specific protein [287-359]
Ligand
BDBM674578
Substrate
n/a
Meas. Tech.
AlphaScreen Assay
IC50
>10000±n/a nM
Citation
 Matzuk, M; Yu, Z; Ku, A; Anglin, J; Li, F; Young, D; Chen, Y; Ucisik, M; Faver, J; Palmer, S; Sharma, R; Kim, C BET SUBFAMILY INHIBITORS AND METHODS USING SAME US Patent  US20240158355 Publication Date 5/16/2024 
Target
Name:
Bromodomain testis-specific protein [287-359]
Synonyms:
BRDT | BRDT_HUMAN | Bromodomain testis-specific protein (BRDT)(BD2)
Type:
n/a
Mol. Mass.:
8713.30
Organism:
Human
Description:
Q58F21[287-359]
Residue:
73
Sequence:
KHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVV
  
Inhibitor
Name:
BDBM674578
Synonyms:
US20240158355, Compound 18
Type:
Small organic molecule
Emp. Form.:
n/a
Mol. Mass.:
n/a
SMILES:
CCn1nc(-c2ccc(N)nc2)c2cc(ccc12)C(=O)Nc1ccc(C)c(NC(C)=O)c1
Structure:
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