Target
Bromodomain testis-specific protein [287-359]
Ligand
BDBM674587
Substrate
n/a
Meas. Tech.
AlphaScreen Assay
IC50
>10000±n/a nM
Citation
 Matzuk, MYu, ZKu, AAnglin, JLi, FYoung, DChen, YUcisik, MFaver, JPalmer, SSharma, RKim, C BET SUBFAMILY INHIBITORS AND METHODS USING SAME US Patent  US20240158355 Publication Date 5/16/2024 
Target
Name:
Bromodomain testis-specific protein [287-359]
Synonyms:
BRDT | BRDT_HUMAN | Bromodomain testis-specific protein (BRDT)(BD2)
Type:
n/a
Mol. Mass.:
8713.30
Organism:
Human
Description:
Q58F21[287-359]
Residue:
73
Sequence:
KHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVV
  
Inhibitor
Name:
BDBM674587
Synonyms:
US20240158355, Compound 27
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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