Reaction Details Report a problem with these data
Target
Bromodomain-containing protein 2 [91-163]
Ligand
BDBM313781
Substrate
n/a
Meas. Tech.
Binding Assay
IC50
550±n/a nM
Citation
 Burns, C; Garnier, J; Sharp, PP; Feutrill, J; Cuzzupe, A Benzodiazepines as bromodomain inhibitors US Patent  US10167292 Publication Date 1/1/2019 
Target
Name:
Bromodomain-containing protein 2 [91-163]
Synonyms:
Bromodomain-containing protein 2 Bromo 1 domain(BRD2 BD1) | Bromodomain-containing protein 2 (BRD2)(BD1) | BRD2_HUMAN | BRD2 | KIAA9001 | RING3
Type:
n/a
Mol. Mass.:
8836.08
Organism:
Human
Description:
BD1 (91-163 aa) of P25440
Residue:
73
Sequence:
WKHQFAWPFRQPVDAVKLGLPDYHKIIKQPMDMGTIKRRLENNYYWAASECMQDFNTMFTNCYIYNKPTDDIV
  
Inhibitor
Name:
BDBM313781
Synonyms:
US10167292, Example 21
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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