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Target
Transcriptional enhancer factor TEF-3 [217-434]
Ligand
BDBM706076
Substrate
n/a
Meas. Tech.
In-Vitro Biochemical TR-FRET Assay
IC50
<1.000±n/a nM
Citation
 CHAPEAU, E; CHENE, P; FURET, P; KIEFFER, L; MACHAUER, R; PICARD, A; SCHMELZLE, T; SELLNER, H; SOLDERMANN, N; VOEGTLE, M; WARTMANN, M BIFUNCTIONAL DEGRADERS COMPRISING A TEAD BINDER US Patent  US20240382600 Publication Date 11/21/2024 
Target
Name:
Transcriptional enhancer factor TEF-3 [217-434]
Synonyms:
Transcriptional enhancer factor TEF-3 (TEAD4)(217-434)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25409.87
Organism:
Human
Description:
Q15561[217-434]
Residue:
218
Sequence:
RSVASSKLWMLEFSAFLEQQQDPDTYNKHLFVHIGQSSPSYSDPYLEAVDIRQIYDKFPEKKGGLKDLFERGPSNAFFLVKFWADLNTNIEDEGSSFYGVSSQYESPENMIITCSTKVCSFGKQVVEKVETEYARYENGHYSYRIHRSPLCEYMINFIHKLKHLPEKYMMNSVLENFTILQVVTNRDTQETLLCIAYVFEVSASEHGAQHHIYRLVKE
  
Inhibitor
Name:
BDBM706076
Synonyms:
US20240382600, Example 5
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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