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Target
Kallikrein-5
Ligand
BDBM33448
Substrate
n/a
Meas. Tech.
Kallikrein 5 1536 HTS Dose Response Confirmation
IC50
2468.02±n/a nM
Citation
 PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Kallikrein-5
Synonyms:
kallikrein-related peptidase 5 preproprotein | KLK5_HUMAN | KLK5 | SCTE | Kallikrein 5
Type:
PROTEIN
Mol. Mass.:
32031.72
Organism:
Human
Description:
EBI_12584
Residue:
293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARSDDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGHYSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPSAGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDSCQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
  
Inhibitor
Name:
BDBM33448
Synonyms:
MLS000527906 | [5-amino-3-(furan-2-yl)-1,2,4-triazol-1-yl]-phenylmethanone | cid_828588 | [5-amino-3-(2-furanyl)-1,2,4-triazol-1-yl]-phenylmethanone | [5-azanyl-3-(furan-2-yl)-1,2,4-triazol-1-yl]-phenyl-methanone | SMR000120480 | (5-Amino-3-furan-2-yl-[1,2,4]triazol-1-yl)-phenyl-methanone | [5-amino-3-(2-furyl)-1,2,4-triazol-1-yl]-phenyl-methanone
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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