Reaction Details
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Report a problem with these dataTarget
cAMP-dependent protein kinase type I-alpha regulatory subunit
Ligand
BDBM51788
Substrate
n/a
Meas. Tech.
Counterscreen for activators of the Protein Kinase A-R2B (PKA-R2B) complex
EC50
>113704±n/a nM
Citation
PubChem, PC Counterscreen for activators of the Protein Kinase A-R2B (PKA-R2B) complex: fluorescence polarization-based biochemical high throughput dose response assay to identify activators of the Protein Kinase A-R1A (PKA-R1A) complex PubChem Bioassay (2011)[AID] More Info.:
Target
Name:
cAMP-dependent protein kinase type I-alpha regulatory subunit
Synonyms:
cAMP-dependent protein kinase | KAP0_BOVIN | PRKAR1A
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42885.14
Organism:
Bovine
Description:
gi_115496662
Residue:
380
Sequence:
MASGTTASEEERSLRECELYVQKHNIQALLKDSIVQLCTARPERPMAFLREYFEKLEKEEAKQIQNLQKAGSRADSREDEISPPPPNPVVKGRRRRGAISAEVYTEEDAASYVRKVIPKDYKTMAALAKAIEKNVLFSHLDDNERSDIFDAMFPVSFIAGETVIQQGDEGDNFYVIDQGEMDVYVNNEWATSVGEGGSFGELALIYGTPRAATVKAKTNVKLWGIDRDSYRRILMGSTLRKRKMYEEFLSKVSILESLDKWERLTVADALEPVQFEDGQKIVVQGEPGDEFFIILEGSAAVLQRRSENEEFVEVGRLGPSDYFGEIALLMNRPRAATVVARGPLKCVKLDRPRFERVLGPCSDILKRNIQQYNSFVSLSV
Inhibitor
Name:
BDBM51788
Synonyms:
cid_5876309 | 5-[(2E)-2-(8-oxidanylidenequinolin-5-ylidene)hydrazinyl]naphthalene-1-sulfonic acid | SMR000555383 | 5-[(2E)-2-(8-oxo-5-quinolinylidene)hydrazinyl]-1-naphthalenesulfonic acid | 5-[(E)-(8-hydroxyquinolin-5-yl)diazenyl]naphthalene-1-sulfonic acid | 5-[(2E)-2-(8-oxoquinolin-5-ylidene)hydrazinyl]naphthalene-1-sulfonic acid | MLS001197249 | 5-[(N'E)-N'-(8-keto-5-quinolylidene)hydrazino]naphthalene-1-sulfonic acid
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
