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Target
Beta-2 adrenergic receptor
Ligand
BDBM50326545
Substrate
n/a
Ki
460±n/a nM
Comments
PDSP_1239
Citation
 Bylund, DB; Snyder, SH Beta adrenergic receptor binding in membrane preparations from mammalian brain. Mol Pharmacol 12:568-80 (1976) [PubMed] 
Target
Name:
Beta-2 adrenergic receptor
Synonyms:
ADRB2_HUMAN | Beta-2 adrenoceptor | ADRB2 | ADRB2R | Beta-2 adrenoreceptor | B2AR
Type:
n/a
Mol. Mass.:
46461.69
Organism:
Human
Description:
P07550
Residue:
413
Sequence:
MGQPGNGSAFLLAPNGSHAPDHDVTQERDEVWVVGMGIVMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGAAHILMKMWTFGNFWCEFWTSIDVLCVTASIETLCVIAVDRYFAITSPFKYQSLLTKNKARVIILMVWIVSGLTSFLPIQMHWYRATHQEAINCYANETCCDFFTNQAYAIASSIVSFYVPLVIMVFVYSRVFQEAKRQLQKIDKSEGRFHVQNLSQVEQDGRTGHGLRRSSKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIQDNLIRKEVYILLNWIGYVNSGFNPLIYCRSPDFRIAFQELLCLRRSSLKAYGNGYSSNGNTGEQSGYHVEQEKENKLLCEDLPGTEDFVGHQGTVPSDNIDSQGRNCSTNDSLL
  
Inhibitor
Name:
BDBM50326545
Synonyms:
CHEMBL1243407 | MJ-9184-1,(+/-) | Zinterol
Type:
Small organic molecule
Emp. Form.:
C19H26N2O4S
Mol. Mass.:
n/a
SMILES:
CC(C)(Cc1ccccc1)NCC(O)c1ccc(O)c(NS(C)(=O)=O)c1
Structure:
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