Reaction Details Report a problem with these data
Target
Acid-sensing ion channel 1
Ligand
BDBM50250132
Substrate
n/a
Meas. Tech.
ChEMBL_1680984 (CHEMBL4031261)
IC50
954993±n/a nM
Citation
More Info.:
Target
Name:
Acid-sensing ion channel 1
Synonyms:
ASIC1_RAT | Accn2 | Acid-sensing ion channel 1 | Amiloride-sensitive cation channel 2, neuronal | Asic1 | Bnac2 | Brain sodium channel 2
Type:
PROTEIN
Mol. Mass.:
59630.33
Organism:
Rattus norvegicus
Description:
ChEMBL_109766
Residue:
526
Sequence:
MELKTEEEEVGGVQPVSIQAFASSSTLHGLAHIFSYERLSLKRALWALCFLGSLAVLLCVCTERVQYYFCYHHVTKLDEVAASQLTFPAVTLCNLNEFRFSQVSKNDLYHAGELLALLNNRYEIPDTQMADEKQLEILQDKANFRSFKPKPFNMREFYDRAGHDIRDMLLSCHFRGEACSAEDFKVVFTRYGKCYTFNSGQDGRPRLKTMKGGTGNGLEIMLDIQQDEYLPVWGETDETSFEAGIKVQIHSQDEPPFIDQLGFGVAPGFQTFVSCQEQRLIYLPSPWGTCNAVTMDSDFFDSYSITACRIDCETRYLVENCNCRMVHMPGDAPYCTPEQYKECADPALDFLVEKDQEYCVCEMPCNLTRYGKELSMVKIPSKASAKYLAKKFNKSEQYIGENILVLDIFFEVLNYETIEQKKAYEIAGLLGDIGGQMGLFIGASILTVLELFDYAYEVIKHRLCRRGKCQKEAKRSSADKGVALSLDDVKRHNPCESLRGHPAGMTYAANILPHHPARGTFEDFTC