Reaction Details Report a problem with these data
Target
Similar to Probable G-protein coupled receptor 92 (Predicted), isoform CRA_a
Ligand
BDBM50454093
Substrate
n/a
Meas. Tech.
ChEMBL_1751827 (CHEMBL4186587)
IC50
>30000±n/a nM
Citation
 Kawamoto, Y; Seo, R; Murai, N; Hiyama, H; Oka, H Identification of potent lysophosphatidic acid receptor 5 (LPA5) antagonists as potential analgesic agents. Bioorg Med Chem 26:257-265 (2018) [PubMed]  Article 
Target
Name:
Similar to Probable G-protein coupled receptor 92 (Predicted), isoform CRA_a
Synonyms:
Lpar5 | Lysophosphatidic acid receptor 5 | Similar to Probable G-protein coupled receptor 92 (Predicted), isoform CRA_a
Type:
PROTEIN
Mol. Mass.:
42940.22
Organism:
Rat
Description:
ChEMBL_117780
Residue:
384
Sequence:
MPQTSFSPHLDAMFANSSANTSSTDSSVPQCRDYRSTHRLHMVVYSLVLATGLPLNALALWVFLRVLRVHSVVSVYMCNLAASDLLFTLSLPLRLSYYARHHWPFPDFLCQTSGAIFQMNMYGSCIFLMLINVDRYAAIVHPLRLRHLRRPLVARRLCLGVWALILLFAVPAARVHSPTTCKYENVTLSLCFESFSDELWKGRLLPLLLLAETLGFLLPLAAVVYSSGRVFWTLARPDATQSHRRQKTVRLLLANLIIFLLCFVPYNSTLAVYGLLRANLVKNSLQARDQVRGVLMIMVLLAGANCVLDPLVYYFSAEGFRNTLRNLGAPFHTRPLPTNGTRGELTEPPSESTQNTGQDATSQRLLQPANLGTRTDNGPQDSAL
  
Inhibitor
Name:
BDBM50454093
Synonyms:
CHEMBL4207356
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
Search PDB for entries with ligand similarity: