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Target
Cytosol aminopeptidase [33-68,L62W]
Ligand
BDBM50457473
Substrate
n/a
Meas. Tech.
ChEMBL_1759783 (CHEMBL4194791)
IC50
30±n/a nM
Citation
 Amin, SA; Adhikari, N; Jha, T Design of Aminopeptidase N Inhibitors as Anti-cancer Agents. J Med Chem 61:6468-6490 (2018) [PubMed]  Article 
Target
Name:
Cytosol aminopeptidase [33-68,L62W]
Synonyms:
Cytosol aminopeptidase | AMPL_PIG | LAP3 | Leucine aminopeptidase (LAP)
Type:
Enzyme
Mol. Mass.:
4015.44
Organism:
Pig
Description:
P28839[33-68,L62W]
Residue:
36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
  
Inhibitor
Name:
BDBM50457473
Synonyms:
CHEMBL4209822
Type:
Small organic molecule
Emp. Form.:
C16H22N2O6
Mol. Mass.:
338.36
SMILES:
CC(C)C[C@@H]([C@H](O)C(=O)NO)C(=O)N[C@H](C(O)=O)c1ccccc1 |r|
Structure:
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