Reaction Details Report a problem with these data
Target
Melatonin receptor type 1B
Ligand
BDBM50495330
Substrate
n/a
Meas. Tech.
ChEMBL_1286910 (CHEMBL3110824)
Ki
26±n/a nM
Citation
 Thireau, J; Marteaux, J; Delagrange, P; Lefoulon, F; Dufourny, L; Guillaumet, G; Suzenet, F Original Design of Fluorescent Ligands by Fusing BODIPY and Melatonin Neurohormone. ACS Med Chem Lett 5:158-61 (2014) [PubMed]  Article 
Target
Name:
Melatonin receptor type 1B
Synonyms:
Mel-1B-R | Mel1b melatonin receptor | Melatonin receptor | Melatonin receptor type 1B | Melatonin 1B | Melatonin receptor type 2 (MT2) | MTR1B_HUMAN | MTNR1B
Type:
Enzyme
Mol. Mass.:
40203.54
Organism:
Human
Description:
P49286
Residue:
362
Sequence:
MSENGSFANCCEAGGWAVRPGWSGAGSARPSRTPRPPWVAPALSAVLIVTTAVDVVGNLLVILSVLRNRKLRNAGNLFLVSLALADLVVAFYPYPLILVAIFYDGWALGEEHCKASAFVMGLSVIGSVFNITAIAINRYCYICHSMAYHRIYRRWHTPLHICLIWLLTVVALLPNFFVGSLEYDPRIYSCTFIQTASTQYTAAVVVIHFLLPIAVVSFCYLRIWVLVLQARRKAKPESRLCLKPSDLRSFLTMFVVFVIFAICWAPLNCIGLAVAINPQEMAPQIPEGLFVTSYLLAYFNSCLNAIVYGLLNQNFRREYKRILLALWNPRHCIQDASKGSHAEGLQSPAPPIIGVQHQADAL
  
Inhibitor
Name:
BDBM50495330
Synonyms:
CHEMBL3109560
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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